SCHEMBL9632474

SCHEMBL9632474

CCOC(=O)N1CCCC(=C(c2ccc(F)cc2)c2ccc(F)cc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
LMNA P02545 3/20 0.49
HRH2 P25021 1/20 0.48
HRH1 P35367 1/20 0.48
HTT P42858 2/20 0.47
RAB9A P51151 1/20 0.47
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
GAA P10253 2/20 0.44
MAPT P10636 2/20 0.44
KDM4E B2RXH2 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
CASP1 P29466 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10601711 0.83 OPRM1 (0.60) ALDH1A1LMNAHRH2HRH1HTT
SCHEMBL4693977 0.81 TSHR (0.57) ALDH1A1LMNAKMT2ACYP2C19L3MBTL1
SCHEMBL9047536 0.80 ALDH1A1 (0.58) ALDH1A1LMNAHRH2HRH1HTT
SCHEMBL5492164 0.78 TSHR (0.51) ALDH1A1LMNAKMT2AL3MBTL1GAA
Carbamic Acid SCHEMBL4082824 0.77 TSHR (0.53) ALDH1A1LMNAKMT2ACYP2C19L3MBTL1
SCHEMBL5496259 0.77 OPRM1 (0.52) ALDH1A1LMNAHTTMEN1KMT2A
SCHEMBL31023851 0.75 ALDH1A1 (0.41) ALDH1A1LMNAKMT2ACYP2C19MAPT
SCHEMBL11319497 0.74 CYP2C19 (0.55) ALDH1A1LMNAHRH2HRH1MEN1
SCHEMBL9872456 0.73 HSD11B1 (0.60) ALDH1A1LMNAHRH2HRH1HTT
SCHEMBL9816191 0.73 DRD2 (0.46) ALDH1A1LMNACYP2C19MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5079249-A Serotine antagonists at 5-HT2 level, antiallergens, antihistamines ADIR ET COMPAGNIE (FR) 1992-01-07 US disclosed
US-5071847-A BIS (ARYL) ALKENE COMPOUNDS OF HOMOPIPERIDINES USEFUL AS SEROTONIN-ANTAGONISTS ADIR ET COMPAGNIE (FR) 1991-12-10 US disclosed
US-5028607-A Antiserotonine agents ADIR ET COMPAGNIE (FR) 1991-07-02 US disclosed