SCHEMBL9633663

SCHEMBL9633663

COC(=O)c1ccc(Cc2cccc3ccc(N(C(C)=O)C4CCCC4)cc23)c(OC)c1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 8/20 0.38
MTNR1B P49286 6/20 0.38
NQO2 P16083 1/20 0.38
NR1H4 Q96RI1 1/20 0.37
C5AR1 P21730 1/20 0.37
DRD2 P14416 1/20 0.37
DRD3 P35462 1/20 0.37
PLA2G4A P47712 2/20 0.37
CYSLTR2 Q9NS75 1/20 0.35
CYSLTR1 Q9Y271 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9633828 0.92 PLA2G4A (0.45) PLA2G4ACYSLTR2CYSLTR1
SCHEMBL9633747 0.84 EPHX2 (0.53) NR1H4PLA2G4ACYSLTR2CYSLTR1
SCHEMBL9825747 0.82 CYSLTR1 (0.48) NR1H4PLA2G4ACYSLTR2CYSLTR1
SCHEMBL9825015 0.80 CYSLTR2 (0.58) PLA2G4ACYSLTR2CYSLTR1
SCHEMBL9634219 0.78 MEN1 (0.35) MTNR1AMTNR1BNQO2CYSLTR2CYSLTR1
SCHEMBL10969445 0.78 KDM4E (0.50) NR1H4
SCHEMBL9634970 0.77 NQO2 (0.49) MTNR1AMTNR1BNQO2PLA2G4A
SCHEMBL9633776 0.77 NQO2 (0.44) MTNR1AMTNR1BNQO2
SCHEMBL9633653 0.77 CYSLTR2 (0.60) CYSLTR2CYSLTR1
SCHEMBL9633804 0.77 NQO2 (0.48) MTNR1AMTNR1BNQO2PLA2G4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0337765-B1 ACYLSULFONAMIDE DERIVATIVES OF ALPHA-CARBOCYCLYLTOLUIC ACIDS USED AS LEUKOTRIENE ANTAGONISTS ICI AMERICAS INC. (US) 1992-10-14 EP disclosed
US-5095038-A Antiinflammatory, antiallergens ICI AMERICAS INC. (US) 1992-03-10 US disclosed
EP-0337765-A2 Acylsulfonamide derivatives of alpha-carbocyclyltoluic acids used as leukotriene antagonists ICI AMERICAS INC. (US) 1989-10-18 EP disclosed