SCHEMBL9636573

SCHEMBL9636573

COCCc1ccc(OC[C@@H]2CN(C(C)C)C(=O)O2)cc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 11/20 0.47
MAPK1 P28482 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NR3C1 P04150 1/20 0.41
ADRB2 P07550 1/20 0.41
ADRB1 P08588 1/20 0.41
CYP2D6 P10635 1/20 0.41
ADRA1A P35348 1/20 0.41
CYP2J2 P51589 1/20 0.41
PDE4D Q08499 1/20 0.41
HTR2B P41595 1/20 0.39
NPY1R P25929 1/20 0.39
NPY2R P49146 1/20 0.39
PMP22 Q01453 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9636582 1.00 GRM2 (0.47) GRM2MAPK1L3MBTL1NR3C1ADRB2
SCHEMBL11161832 0.84 GRM2 (0.50) GRM2MAPK1L3MBTL1HTR2B
SCHEMBL11160325 0.83 GRM2 (0.62) GRM2MAPK1L3MBTL1HTR2BNPSR1
SCHEMBL24933695 0.82 GRM2 (0.51) GRM2MAPK1L3MBTL1CYP2D6HTR2B
SCHEMBL3372293 0.81 GRM2 (0.63) GRM2MAPK1L3MBTL1HTR2BTDP1
SCHEMBL11154054 0.80 ADRB2 (0.45) GRM2MAPK1L3MBTL1ADRB2ADRB1
SCHEMBL7909523 0.80 GRM2 (0.49) GRM2MAPK1L3MBTL1HTR2B
SCHEMBL11154145 0.76 GRM2 (0.46) GRM2MAPK1L3MBTL1HTR2B
SCHEMBL4902039 0.75 ALDH1A1 (0.57) NR3C1ADRB2ADRB1CYP2D6ADRA1A
SCHEMBL4081261 0.75 ALDH1A1 (0.57) NR3C1ADRB2ADRB1CYP2D6ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013141437-A1 METHOD FOR MANUFACTURING HIGH PURITY (S)-METOPROLOL 주식회사 알에스텍 (KR) 2013-09-26 WO disclosed
EP-0339006-B1 PROCESS FOR PREPARING S-METOPROLOL AND INTERMEDIATES THEREFOR Astra Pharmaceutical Production AB (SE) 1992-07-08 EP disclosed
US-5034535-A Multistage reaction with chloroformate ester and isopropylamino-1,2-propanediol for cyclization, sulfonation and etherification ASTRA PHARMACEUTICAL PRODUCTION AKTIEBOLAG (SE) 1991-07-23 US disclosed
EP-0339006-A1 Process for preparing S-metoprolol and intermediates therefor Astra Pharmaceutical Production AB (SE) 1989-10-25 EP disclosed