SCHEMBL966252

SCHEMBL966252

CCOC(=O)CNS(=O)(=O)NC(=O)OC(C)(C)C

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.74
CA14 Q9ULX7 4/20 0.74
CA2 P00918 1/20 0.74
CA1 P00915 2/20 0.50
CA7 P43166 2/20 0.50
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
HTT P42858 1/20 0.42
CTSK P43235 1/20 0.39
GAA P10253 2/20 0.39
MGAM O43451 1/20 0.38
SI P14410 1/20 0.38
MGAM2 Q2M2H8 1/20 0.38
ALDH1A1 P00352 3/20 0.36
MEN1 O00255 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36
KDM4E B2RXH2 1/20 0.36
PKM P14618 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22398321 0.87 CA12 (0.84) CA12CA14CA2CA1CA7
SCHEMBL4442641 0.80 CA12 (0.73) CA12CA14CA2CA1CA7
SCHEMBL13966219 0.80 CA12 (0.67) CA12CA14CA2CA1CA7
SCHEMBL12959650 0.80 GAA (0.46) CA12CA14CA2CYP1A2GAA
SCHEMBL8066895 0.78 CA1 (0.68) CA12CA14CA2CA1CA7
SCHEMBL1936376 0.78 ALDH1A1 (0.52) CA12CA14CA2CA1CYP1A2
SCHEMBL3295077 0.77 CA12 (0.44) CA12CA14CA2GAAMGAM
SCHEMBL20646495 0.77 CA12 (0.63) CA12CA14CA2CA1CA7
SCHEMBL22404346 0.75 CA12 (0.56) CA12CA14CA2CA1CA7
SCHEMBL16472070 0.75 CA12 (0.65) CA12CA14CA2CA1CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 75 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109810104-B Method for synthesizing indoleamine 2, 3-dioxygenase inhibitors 因赛特控股公司 2022-05-03 CN disclosed
EP-3744715-A1 PROCESS FOR THE SYNTHESIS OF AN INDOLEAMINE 2,3-DIOXYGENASE INHIBITOR Incyte Holdings Corporation (US) 2020-12-02 EP disclosed
EP-3744715-A1 PROCESS FOR THE SYNTHESIS OF AN INDOLEAMINE 2,3-DIOXYGENASE INHIBITOR Incyte Holdings Corporation (US) 2020-12-02 EP disclosed
EP-3066085-B1 PROCESS FOR THE SYNTHESIS OF AN INDOLEAMINE 2,3-DIOXYGENASE INHIBITOR INCYTE HOLDINGS CORP (US) 2020-05-13 EP disclosed
EP-3066085-B1 PROCESS FOR THE SYNTHESIS OF AN INDOLEAMINE 2,3-DIOXYGENASE INHIBITOR INCYTE HOLDINGS CORP (US) 2020-05-13 EP disclosed
CN-109810104-A Method for synthesis of indole amine 2,3- dioxygenase inhibitor 因赛特控股公司 2019-05-28 CN disclosed
US-10280157-B2 Process for the synthesis of an indoleamine 2,3-dioxygenase inhibitor INCYTE CORPORATION (US) 2019-05-07 US disclosed
US-10280157-B2 Process for the synthesis of an indoleamine 2,3-dioxygenase inhibitor INCYTE CORPORATION (US) 2019-05-07 US disclosed
CN-105899498-B Method for synthesizing indoleamine 2, 3-dioxygenase inhibitors 因赛特控股公司 2019-01-25 CN disclosed
US-20180319812-A1 HETEROCYCLIC COMPOUND ACTION MEDICAL TECHNOLOGIES, LLC 2018-11-08 US disclosed
US-20080045706-A1 Anti-inflammatory medicaments DECIPHERA PHARMACEUTICALS, LLC 2008-02-21 US disclosed
US-20080045531-A1 Anti-inflammatory medicaments DECIPHERA PHARMACEUTICALS, LLC 2008-02-21 US disclosed
US-7279576-B2 Anti-cancer medicaments DECIPHERA PHARMACEUTICALS, LLC (US) 2007-10-09 US disclosed
US-7279576-B2 Anti-cancer medicaments DECIPHERA PHARMACEUTICALS, LLC (US) 2007-10-09 US disclosed
US-20070191336-A1 p38 kinase inhibitors DECIPHERA PHARMACEUTICALS, LLC 2007-08-16 US disclosed
US-20070191336-A1 p38 kinase inhibitors DECIPHERA PHARMACEUTICALS, LLC 2007-08-16 US disclosed
US-7202257-B2 Anti-inflammatory medicaments DECIPHERA PHARMACEUTICALS, LLC (US) 2007-04-10 US disclosed
US-7202257-B2 Anti-inflammatory medicaments DECIPHERA PHARMACEUTICALS, LLC (US) 2007-04-10 US disclosed
US-20070037808-A1 p38 kinase inhibitors DECIPHERA PHARMACEUTICALS, LLC 2007-02-15 US disclosed
US-20070037808-A1 p38 kinase inhibitors DECIPHERA PHARMACEUTICALS, LLC 2007-02-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080045706-A1 Anti-inflammatory medicaments MIF, PTGES2, TNF CA12 2354/4885CA14 3053/4885CA2 860/4885
US-20070037808-A1 p38 kinase inhibitors MAPK1, MAP3K8, MAP3K1 CA12 4553/4885CA14 4756/4885CA2 3205/4885
US-20180319812-A1 HETEROCYCLIC COMPOUND RORC, RORB, RORA CA12 1747/4885CA14 2343/4885CA2 857/4885
US-20080045531-A1 Anti-inflammatory medicaments MIF, PTGES2, TNF CA12 2354/4885CA14 3053/4885CA2 860/4885
US-20070191336-A1 p38 kinase inhibitors MAPK1, MAP3K8, MAP3K1 CA12 4553/4885CA14 4756/4885CA2 3205/4885
US-10280157-B2 Process for the synthesis of an indoleamine 2,3-dioxygenase inhibitor IDO1, INMT, IDO2 CA12 3758/4885CA14 3477/4885CA2 1698/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.