SCHEMBL9665356

SCHEMBL9665356

CCN1C(=O)C(C(=O)Nc2ccc(F)cc2F)c2cc(C(C)=O)ccc21

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
HSD17B10 Q99714 1/20 0.40
GAA P10253 1/20 0.40
PKM P14618 2/20 0.40
TP53 P04637 1/20 0.40
ATM Q13315 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9665452 0.90 MAPT (0.48) MAPTSMN1; SMN2L3MBTL1KMT2AMEN1
SCHEMBL9665440 0.88 TP53 (0.44) SMN1; SMN2L3MBTL1KMT2ATP53ATM
SCHEMBL9667871 0.88 TP53 (0.44) MAPTL3MBTL1KMT2AMEN1HSD17B10
SCHEMBL10737485 0.84 MEN1 (0.41) MAPTSMN1; SMN2KMT2AMEN1HSD17B10
SCHEMBL9666166 0.82 L3MBTL1 (0.43) MAPTL3MBTL1KMT2AMEN1HSD17B10
SCHEMBL10738159 0.81 MAPT (0.44) MAPTSMN1; SMN2KMT2AMEN1HSD17B10
SCHEMBL10733852 0.79 PTGS2 (0.42) MAPTL3MBTL1KMT2AMEN1HSD17B10
SCHEMBL9667449 0.77 MEN1 (0.46) MAPTSMN1; SMN2KMT2AMEN1GAA
SCHEMBL7234484 0.77 ALDH1A1 (0.45) MAPTKMT2AMEN1GAAPOLB
SCHEMBL10732971 0.76 ALDH1A1 (0.42) MAPTSMN1; SMN2L3MBTL1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0181136-B1 OXINDOLE ANTIINFLAMMATORY AGENTS PFIZER INC. (US) 1992-03-25 EP disclosed
US-4686224-A Oxindole antiinflammatory agents PFIZER INC. (US) 1987-08-11 US disclosed
US-4644005-A ANTIARTHRITIC AGENTS PFIZER INC. (US) 1987-02-17 US disclosed
EP-0181136-A2 Oxindole antiinflammatory agents PFIZER INC. (US) 1986-05-14 EP disclosed