SCHEMBL9681952

SCHEMBL9681952

Fc1ccc(-n2nc(N3CCN(CC4CC4)CC3)c3ccccc32)cc1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.45
HTR1A P08908 3/20 0.40
HTR2C P28335 2/20 0.40
DRD2 P14416 3/20 0.39
DRD3 P35462 3/20 0.39
HTR2A P28223 1/20 0.39
SMO Q99835 1/20 0.39
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
HTR3A P46098 1/20 0.39
HTR3D Q70Z44 1/20 0.39
HTR3C Q8WXA8 1/20 0.39
CYP17A1 P05093 1/20 0.39
CYP21A2 P08686 1/20 0.39
CYP11B1 P15538 1/20 0.39
MAPT P10636 1/20 0.38
PARP1 P09874 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9680782 0.99 LMNA (0.44) LMNAHTR1AHTR2CDRD2DRD3
SCHEMBL9682466 0.90 DRD3 (0.47) LMNAHTR1AHTR2CDRD2DRD3
SCHEMBL9680355 0.88 SLC6A2 (0.44) HTR1AHTR2CDRD2DRD3HTR2A
SCHEMBL9763064 0.84 KHK (0.51) LMNASMO
Hydrochloric Acid SCHEMBL9681944 0.83 KHK (0.50) LMNASMO
SCHEMBL9681232 0.81 HTR1A (0.44) LMNAHTR1AHTR2CSMOHTR3E
Bromide SCHEMBL9681411 0.81 HTR1A (0.44) LMNAHTR1AHTR2CSMOHTR3E
SCHEMBL9681940 0.80 KHK (0.48) LMNAHTR1AHTR2CHTR3EHTR3B
SCHEMBL9681305 0.78 KHK (0.47) HTR1AHTR2CHTR3AMAPT
SCHEMBL9680606 0.75 TP53 (0.45) LMNASMOMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US claimed
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed