SCHEMBL9683244

SCHEMBL9683244

FC(F)(F)c1ccc(-n2nc(N3CCN(CCc4ccccc4)CC3)c3ccccc32)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.54
ADRA1D P25100 1/20 0.49
ADRA1A P35348 1/20 0.49
ADRA1B P35368 1/20 0.49
MAPT P10636 3/20 0.47
ALDH1A1 P00352 2/20 0.47
MAPK1 P28482 2/20 0.47
LMNA P02545 1/20 0.47
POLB P06746 1/20 0.47
HSD17B10 Q99714 1/20 0.47
HTR1A P08908 2/20 0.47
DRD2 P14416 1/20 0.47
SLC6A2 P23975 1/20 0.47
SLC6A4 P31645 1/20 0.47
NPSR1 Q6W5P4 1/20 0.45
DRD4 P21917 1/20 0.43
GRM2 Q14416 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9681380 0.99 SIGMAR1 (0.53) SIGMAR1ADRA1DADRA1AADRA1BMAPT
SCHEMBL9681250 0.89 HTR1A (0.60) SIGMAR1MAPTALDH1A1MAPK1LMNA
SCHEMBL9680665 0.88 MAPK1 (0.46) ADRA1DADRA1AADRA1BMAPTALDH1A1
SCHEMBL9763384 0.85 KHK (0.48) MAPTALDH1A1LMNADRD4GRM2
SCHEMBL9680624 0.84 CYP1A2 (0.46) MAPTMAPK1LMNAHSD17B10HTR1A
SCHEMBL9680355 0.83 SLC6A2 (0.44) MAPTHTR1ADRD2SLC6A2SLC6A4
Fumaric Acid SCHEMBL9681243 0.80 KHK (0.44) ALDH1A1MAPK1LMNADRD4GRM2
Fumaric Acid SCHEMBL9681235 0.80 KHK (0.44) ALDH1A1MAPK1LMNADRD4GRM2
SCHEMBL9682489 0.79 HTR6 (0.47) SIGMAR1MAPTALDH1A1HTR1ANPSR1
Hydrochloric Acid SCHEMBL9680573 0.78 HTR6 (0.46) SIGMAR1MAPTALDH1A1HTR1ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US claimed
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed