SCHEMBL9682463

SCHEMBL9682463

COC(=O)OC[C@H]1O[C@@H](n2cnc3c(OC)nc(N)nc32)[C@H](OC(=S)Oc2ccccc2)[C@H]1OS(C)(=O)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HINT1 P49773 3/20 0.42
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ADORA3 P0DMS8 3/20 0.38
ADORA2A P29274 3/20 0.38
ADORA2B P29275 3/20 0.38
ADORA1 P30542 2/20 0.38
ACHE P22303 2/20 0.36
PRKAB2 O43741 1/20 0.35
PRKAG1 P54619 1/20 0.35
PRKAA2 P54646 1/20 0.35
PRKAA1 Q13131 1/20 0.35
PRKAG3 Q9UGI9 1/20 0.35
PRKAG2 Q9UGJ0 1/20 0.35
PRKAB1 Q9Y478 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9681390 0.84 HINT1 (0.51) HINT1ADORA3ADORA2AADORA2BADORA1
SCHEMBL9680659 0.81 PNP (0.37) HINT1ALDH1A1LMNATP53MAPT
SCHEMBL9683196 0.75 P2RY1 (0.40) HINT1
SCHEMBL9683203 0.75 P2RY1 (0.40) HINT1
SCHEMBL8527967 0.74 ALDH1A1 (0.66) HINT1ALDH1A1LMNATP53MAPT
SCHEMBL9682513 0.74 ACHE (0.48) HINT1ALDH1A1LMNATP53MAPT
SCHEMBL10444503 0.72 LMNA (0.45) HINT1ALDH1A1LMNATP53MAPT
SCHEMBL9681406 0.71 HINT1 (0.42) HINT1ADORA3ADORA2AADORA2BADORA1
SCHEMBL8531895 0.70 ALDH1A1 (0.57) HINT1ALDH1A1LMNATP53MAPT
SCHEMBL8532634 0.70 ALDH1A1 (0.57) HINT1ALDH1A1LMNATP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5153318-A Viricides for hepatitis and human t-cell leukemia/lymphoma viruses BURROUGHS WELLCOME CO. (US) 1992-10-06 US disclosed
EP-0421739-A1 3'-azido purine nucleoside THE WELLCOME FOUNDATION LIMITED (GB) 1991-04-10 EP disclosed