SCHEMBL9682813

SCHEMBL9682813

Cn1cccc(C2=CC(C)(C)Oc3ccc(C#N)cc32)c1=O

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
ABCC9 O60706 7/20 0.36
ABCC8 Q09428 3/20 0.36
KCNJ11 Q14654 3/20 0.36
KCNJ8 Q15842 3/20 0.36
ABCB1 P08183 7/20 0.35
CASP3 P42574 1/20 0.35
MALT1 Q9UDY8 1/20 0.34
HTR2A P28223 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9680361 0.86 KDM4E (0.36) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL9680894 0.82 RARA (0.33) MALT1
SCHEMBL9681489 0.82 ALDH1A1 (0.41) ABCB1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL9682156 0.80 ALDH1A1 (0.38) CASP3MALT1
SCHEMBL9682834 0.78 PDPK1 (0.39) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL9525977 0.77 OPRD1 (0.37) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL9680331 0.77 RARA (0.40) CASP3LMNA
SCHEMBL8195282 0.75 OPRD1 (0.44) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL9523959 0.75 PDE4A (0.37) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL9527583 0.75 PDE4A (0.42) PDE4APDE4BPDE4CPDE4DABCC9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112839-A CHROMAN DERIVATIVES MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-05-12 US disclosed