SCHEMBL9680331

SCHEMBL9680331

COC(=O)c1ccc2c(c1)C(c1cccn(C)c1=O)=CC(C)(C)O2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 2/20 0.40
RARB P10826 2/20 0.40
RARG P13631 2/20 0.40
CASP3 P42574 1/20 0.39
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
KCNH2 Q12809 1/20 0.37
ALOX5 P09917 1/20 0.37
RAB9A P51151 4/20 0.36
SMN1; SMN2 Q16637 4/20 0.36
MAPT P10636 3/20 0.36
NPC1 O15118 2/20 0.36
PDK2 Q15119 2/20 0.36
PKM P14618 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9680402 0.87 RARA (0.39) RARARARBRARGCASP3OPRD1
SCHEMBL9681433 0.83 CFTR (0.42) RARARARBRARGMAPTMEN1
SCHEMBL12365911 0.81 RARA (0.43) RARARARBRARGOPRD1OPRK1
SCHEMBL2263334 0.80 RARA (0.43) RARARARBRARGOPRD1OPRK1
SCHEMBL12365916 0.80 NPC1 (0.44) RARARARBRARGOPRD1OPRK1
SCHEMBL9680894 0.80 RARA (0.33) RARARARBRARGRAB9AMAPT
SCHEMBL9680947 0.80 PDPK1 (0.43) RARARARBRARGCASP3OPRD1
SCHEMBL12365140 0.78 RARA (0.55) RARARARBRARGCASP3OPRD1
SCHEMBL9682813 0.77 PDE4A (0.37) CASP3LMNA
SCHEMBL9682156 0.77 ALDH1A1 (0.38) CASP3RAB9ANPC1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112839-A CHROMAN DERIVATIVES MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-05-12 US disclosed