SCHEMBL9684657

SCHEMBL9684657

C[C@@H](N)C(=O)NC1CCN1C(c1ccccc1)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 8/20 0.45
OPRD1 P41143 8/20 0.45
OPRK1 P41145 8/20 0.45
OPRL1 P41146 8/20 0.45
XIAP P98170 5/20 0.45
HTT P42858 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
GAA P10253 1/20 0.43
CTRB1 P17538 2/20 0.42
KMT2A Q03164 1/20 0.41
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6025516 0.75 OPRM1 (0.48) OPRM1OPRD1OPRK1OPRL1KMT2A
SCHEMBL2770710 0.69 KMT2A (0.48) OPRM1OPRD1OPRK1OPRL1KMT2A
SCHEMBL5685739 0.68 ALDH1A1 (0.47) OPRM1OPRD1OPRK1OPRL1HTT
SCHEMBL5685826 0.68 ALDH1A1 (0.47) OPRM1OPRD1OPRK1OPRL1HTT
SCHEMBL5685743 0.68 ALDH1A1 (0.47) OPRM1OPRD1OPRK1OPRL1HTT
SCHEMBL10783873 0.68 OPRM1 (0.46) OPRM1OPRD1OPRK1OPRL1HTT
SCHEMBL4848461 0.67 SIGMAR1 (0.65) KMT2A
SCHEMBL9194851 0.66 CTSD (0.58) HTTNPSR1GAACTRB1KMT2A
SCHEMBL9194859 0.66 CTSD (0.58) HTTNPSR1GAACTRB1KMT2A
SCHEMBL29046178 0.66 OPRM1 (0.42) OPRM1OPRD1OPRK1OPRL1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0514268-A1 Substituted amino acid azetidinyl pyridone derivatives, their preparation and use as medicines LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 1992-11-19 EP disclosed