[11C]Sa4503

[11C]Sa4503

SCHEMBL968642

COc1ccc(CCN2CCN(CCCc3ccccc3)CC2)cc1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 1.00
EBP Q15125 2/20 1.00
TMEM97 Q5BJF2 1/20 1.00
EBPL Q9BY08 1/20 0.86
ABCB1 P08183 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
[11C]Sa4503 SCHEMBL29358558 1.00 SIGMAR1 (1.00) SIGMAR1EBPTMEM97EBPLABCB1
[11C]Sa4503 SCHEMBL29358694 0.99 SIGMAR1 (0.97) SIGMAR1EBPTMEM97EBPLABCB1
[11C]Sa4503 SCHEMBL1299046 0.99 SIGMAR1 (0.97) SIGMAR1EBPTMEM97EBPLABCB1
Hydrochloric Acid SCHEMBL8088187 0.99 SIGMAR1 (0.97) SIGMAR1EBPTMEM97EBPLABCB1
SCHEMBL8083210 0.97 SIGMAR1 (0.95) SIGMAR1EBPTMEM97EBPLABCB1
SCHEMBL8086559 0.96 SIGMAR1 (0.92) SIGMAR1EBPTMEM97EBPLABCB1
Hydrochloric Acid SCHEMBL8075024 0.96 SIGMAR1 (0.92) SIGMAR1EBPTMEM97EBPLABCB1
Hydrochloric Acid SCHEMBL8086545 0.95 SIGMAR1 (0.90) SIGMAR1EBPTMEM97EBPLABCB1
SCHEMBL8075010 0.94 SIGMAR1 (0.89) SIGMAR1EBPTMEM97EBPL
Hydrochloric Acid SCHEMBL8074974 0.94 SIGMAR1 (0.88) SIGMAR1EBPTMEM97EBPLABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 157 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116981449-A Compounds and compositions for inducing neuroprotection 瑞斯特医疗公司 2023-10-31 CN claimed
EP-4142703-B1 COMPOUND AND COMPOSITION FOR INDUCING NEUROPROTECTION REST THERAPEUTICS (FR) 2023-10-18 EP claimed
US-20230270695-A1 COMPOUND AND COMPOSITION FOR INDUCING NEUROPROTECTION INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 2023-08-31 US claimed
EP-4142703-A1 COMPOUND AND COMPOSITION FOR INDUCING NEUROPROTECTION REST THERAPEUTICS (FR) 2023-03-08 EP claimed
WO-2021234324-A1 COMPOUND AND COMPOSITION FOR INDUCING NEUROPROTECTION REST THERAPEUTICS (FR) 2021-11-25 WO claimed
EP-3880209-A1 COMPOSITIONS AND METHODS FOR REGULATING INFLAMMATION University of Virginia Patent Foundation (US) 2021-09-22 EP claimed
EP-3104847-B1 NOVEL USE OF SIGMA-1 RECEPTOR AGONIST COMPOUNDS MTA TAMOGATOTT KUTATOCSOPORTOK IRODAJA (HU) 2020-11-11 EP claimed
WO-2020118086-A1 COMPOSITIONS AND METHODS FOR REGULATING INFLAMMATION UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2020-06-11 WO claimed
CN-106456578-B Use of SIGMA-1 receptor agonist compounds 匈牙利科学院大学及其他机构附属研究所 2020-02-18 CN claimed
CN-106456578-A Novel use of SIGMA-1 receptor agonist compounds 匈牙利科学院大学及其他机构附属研究所 2017-02-22 CN claimed
WO-2015118365-A1 NOVEL USE OF SIGMA-1 RECEPTOR AGONIST COMPOUNDS MTA TÁMOGATOTT KUTATÓCSOPORTOK IRODÁJA (HU) 2015-08-13 WO claimed
US-20110152284-A1 Sigma ligands for neuronal regeneration and functional recovery WIELOCH TADEUSZ 2011-06-23 US claimed
US-20110015209-A1 Sigma ligands for neuronal regeneration and functional recovery M'S SCIENCE CORPORATION 2011-01-20 US claimed
US-7863272-B2 Sigma ligands for neuronal regeneration and functional recovery M'S SCIENCE CORPORATION (JP) 2011-01-04 US claimed
US-7829562-B2 Sigma ligands for neuronal regeneration and functional recovery M'S SCIENCE CORPORATION (JP) 2010-11-09 US claimed
WO-2008060271-A1 SIGMA LIGANDS FOR NEURONAL REGENERATION AND FUNCTIONAL RECOVERY M'S SCIENCE CORPORATION (JP) 2008-05-22 WO claimed
US-6436938-B1 ADMINISTERING A SIGMA RECEPTOR LIGAND IN COMBINATION WITH AN ANTIDEPRESSANT AGENT; ESPECIALLY FOR REFRACTORY DEPRESSION PFIZER INC. 2002-08-20 US claimed
US-20020099045-A1 Combination treatment for depression PFIZER PRODUCTS INC. 2002-07-25 US claimed
EP-1224930-A1 Combination of a SR inhibitor and sigma receptor ligand in the treatment ofdepression Pfizer Products Inc. (US) 2002-07-24 EP claimed
WO-2002030422-A1 USE OF DEFINED SUBSTANCES THAT BIND TO THE SIGMA RECEPTOR FOR COMBATING SARCOMA AND CARCINOMA MERCK PATENT GMBH (DE) 2002-04-18 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110152284-A1 Sigma ligands for neuronal regeneration and functional recovery SIGMAR1, TMEM97, LPAR6 SIGMAR1 1/4885EBP 894/4885TMEM97 2/4885
US-20230270695-A1 COMPOUND AND COMPOSITION FOR INDUCING NEUROPROTECTION BDNF, GAP43, NLN SIGMAR1 1214/4885EBP 68/4885TMEM97 1922/4885
US-20110015209-A1 Sigma ligands for neuronal regeneration and functional recovery SIGMAR1, TMEM97, GPR6 SIGMAR1 1/4885EBP 979/4885TMEM97 2/4885
US-20020099045-A1 Combination treatment for depression HTR5A, HTR1A, OPRL1 SIGMAR1 13/4885EBP 1526/4885TMEM97 50/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.