SCHEMBL9687000

SCHEMBL9687000

COc1cc(C=O)cc(C(=O)[O-])c1O.COc1cc(C=O)cc(C(=O)[O-])c1O.[Ca+2]

nearest known ligand 0.50

Known targets — ChEMBL curated mechanism

GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHMGCRMMP1MMP13MMP7MMP8PTGS1PTGS2ileSpolrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 known ✓ P23219 2/20 0.49
PTGS2 known ✓ P35354 1/20 0.49
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2B6 P20813 1/20 0.50
PKM P14618 1/20 0.49
ALDH1A1 P00352 4/20 0.47
HPGD P15428 2/20 0.47
TRIM24 O15164 1/20 0.47
ALDH5A1 P51649 1/20 0.47
ABAT P80404 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
TRIM33 Q9UPN9 1/20 0.47
ALOX5 P09917 3/20 0.44
STAT3 P40763 2/20 0.44
NFE2L2 Q16236 2/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Potassium Ion SCHEMBL9688312 0.97 ALDH1A1 (0.47) CYP1A2CYP3A4CYP2D6CYP2C9CYP2B6
SCHEMBL9686348 0.97 ALDH1A1 (0.47) CYP1A2CYP3A4CYP2D6CYP2C9CYP2B6
SCHEMBL9686330 0.97 ALDH1A1 (0.47) CYP1A2CYP3A4CYP2D6CYP2C9CYP2B6
SCHEMBL29954196 0.83 PKM (0.51) CYP1A2CYP3A4CYP2D6CYP2C9CYP2B6
SCHEMBL1981806 0.83 PKM (0.51) CYP1A2CYP3A4CYP2D6CYP2C9CYP2B6
SCHEMBL9687016 0.83 KDM4E (0.55) CYP1A2CYP3A4ALDH1A1HPGDGAA
SCHEMBL4757716 0.82 KMT2A (0.49) CYP1A2CYP3A4CYP2D6CYP2C9CYP2B6
SCHEMBL4756891 0.82 ALDH1A1 (0.49) CYP1A2CYP3A4CYP2D6CYP2C9CYP2B6
SCHEMBL9686354 0.82 PKM (0.50) CYP1A2CYP3A4CYP2D6CYP2C9CYP2B6
SCHEMBL9687007 0.82 PKM (0.50) CYP1A2CYP3A4CYP2D6CYP2C9CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0514202-A2 Smoking compositions containing a vanillin-release additive Philip Morris Products Inc. (US) 1992-11-19 EP claimed
US-5144965-A Vanillin carboxylate type additive pyrolyzes to ethyl vanillin; cigarettes PHILIP MORRIS INCORPORATED (US) 1992-09-08 US claimed
EP-0514202-A2 Smoking compositions containing a vanillin-release additive Philip Morris Products Inc. (US) 1992-11-19 EP disclosed
US-5144965-A Vanillin carboxylate type additive pyrolyzes to ethyl vanillin; cigarettes PHILIP MORRIS INCORPORATED (US) 1992-09-08 US disclosed