SCHEMBL9688183

SCHEMBL9688183

N#Cc1ccccc1OCC(O)CNCCc1nc2cc(-c3ccc(=O)[nH]n3)ccc2[nH]1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.48
ADRB1 P08588 15/20 0.43
ADRB2 P07550 1/20 0.43
ADRB3 P13945 1/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
ALOX15 P16050 1/20 0.43
KMT2A Q03164 1/20 0.43
CASR P41180 1/20 0.42
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9688229 0.94 CTSS (0.48) CTSSADRB1ADRB2ADRB3KDM4E
SCHEMBL9687230 0.88 MAPK1 (0.45) ADRB1ADRB2ADRB3CYP1A2CYP2D6
SCHEMBL7303647 0.82 CTSS (0.45) CTSSADRB1ADRB2ADRB3KDM4E
SCHEMBL7303996 0.80 CTSS (0.43) CTSSADRB1ADRB2ADRB3KDM4E
SCHEMBL7303661 0.76 CTSS (0.45) CTSSADRB1ADRB2ADRB3KDM4E
SCHEMBL7304010 0.74 PDE3B (0.43) CTSSADRB1ADRB2ADRB3KDM4E
SCHEMBL9687213 0.70 MAPK1 (0.44) ADRB1ADRB2ADRB3MEN1CYP1A2
SCHEMBL11803062 0.70 ADRB1 (0.72) ADRB1ADRB2ADRB3KDM4EMEN1
SCHEMBL7306568 0.69 ADRB2 (0.39) ADRB1ADRB2ADRB3KDM4ECYP1A2
SCHEMBL7303724 0.68 RAD52 (0.43) KDM4EMEN1CYP1A2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135932-A 2-HYDROXYPROPYLAMINO-ALKYL-BENZIMIDAZOLY-5-YL DERIVATIVES AND THEIR USE IN THE TREATMENT OF HEART DISEASE DR. KARL THOMAE GMBH (DE) 1992-08-04 US disclosed