SCHEMBL9687230

SCHEMBL9687230

O=c1ccc(-c2ccc3[nH]c(CCNCC(O)COc4cccc5ccccc45)nc3c2)n[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
HTT P42858 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
ADRB1 P08588 7/20 0.41
ADRB2 P07550 9/20 0.41
CYP2D6 P10635 4/20 0.40
SIGMAR1 Q99720 4/20 0.39
ADRB3 P13945 4/20 0.39
CYP1A2 P05177 3/20 0.39
SLC6A4 P31645 3/20 0.39
HTR2B P41595 3/20 0.39
NR2E1 Q9Y466 3/20 0.39
ALDH1A1 P00352 3/20 0.39
HTR2A P28223 3/20 0.39
HTR2C P28335 3/20 0.39
HTR6 P50406 3/20 0.39
SCN1A P35498 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9688183 0.88 CTSS (0.48) ADRB1ADRB2CYP2D6ADRB3CYP1A2
SCHEMBL9688229 0.81 CTSS (0.48) ADRB1ADRB2ADRB3CYP1A2
SCHEMBL9687213 0.81 MAPK1 (0.44) MAPK1SMN1; SMN2GAAMAPTHTT
SCHEMBL9687447 0.79 MAPK1 (0.41) MAPK1SMN1; SMN2GAAMAPTHTT
SCHEMBL9687223 0.77 PIK3CA (0.34) HTTCYP2C9
SCHEMBL7304449 0.75 PDE3B (0.39) MAPK1SMN1; SMN2GAAMAPTHTT
SCHEMBL7306568 0.70 ADRB2 (0.39) MAPK1GAAMAPTADRB1ADRB2
SCHEMBL7303647 0.70 CTSS (0.45) ADRB1ADRB2ADRB3CYP1A2
SCHEMBL7303724 0.69 RAD52 (0.43) MAPK1SMN1; SMN2MAPTCYP1A2LMNA
SCHEMBL4845731 0.66 ADRB2 (0.67) MAPK1SMN1; SMN2GAAMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135932-A 2-HYDROXYPROPYLAMINO-ALKYL-BENZIMIDAZOLY-5-YL DERIVATIVES AND THEIR USE IN THE TREATMENT OF HEART DISEASE DR. KARL THOMAE GMBH (DE) 1992-08-04 US disclosed