SCHEMBL9687213

SCHEMBL9687213

O=C1CCC(c2ccc3[nH]c(CCNCC(O)COc4cccc5ccccc45)nc3c2)=NN1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
ADRB1 P08588 7/20 0.40
ADRB2 P07550 8/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP1A2 P05177 3/20 0.38
CYP2D6 P10635 3/20 0.38
SLC6A4 P31645 3/20 0.38
HTR2B P41595 3/20 0.38
SIGMAR1 Q99720 3/20 0.38
NR2E1 Q9Y466 3/20 0.38
ADRB3 P13945 3/20 0.38
ALDH1A1 P00352 2/20 0.38
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303647 0.88 CTSS (0.45) ADRB1ADRB2MEN1KMT2ACYP1A2
SCHEMBL7306568 0.88 ADRB2 (0.39) MAPK1GAAMAPTADRB1ADRB2
SCHEMBL9687447 0.85 MAPK1 (0.41) MAPK1SMN1; SMN2GAAMAPTHTT
SCHEMBL7302924 0.84 MEN1 (0.39) SMN1; SMN2NPSR1ADRB1MEN1KMT2A
SCHEMBL7306574 0.82 ADRB2 (0.39) MAPK1GAAMAPTADRB1ADRB2
SCHEMBL7303661 0.82 CTSS (0.45) ADRB1ADRB2MEN1KMT2ACYP1A2
SCHEMBL9687230 0.81 MAPK1 (0.45) MAPK1SMN1; SMN2GAAMAPTHTT
SCHEMBL7304449 0.81 PDE3B (0.39) MAPK1SMN1; SMN2GAAMAPTHTT
SCHEMBL7302583 0.79 MAPT (0.42) MAPTADRB1ADRB2KMT2AADRB3
SCHEMBL9687567 0.78 KMT2A (0.39) SMN1; SMN2NPSR1MEN1KMT2AADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135932-A 2-HYDROXYPROPYLAMINO-ALKYL-BENZIMIDAZOLY-5-YL DERIVATIVES AND THEIR USE IN THE TREATMENT OF HEART DISEASE DR. KARL THOMAE GMBH (DE) 1992-08-04 US disclosed