SCHEMBL9689430

SCHEMBL9689430

COC(=O)OC1=C(C)NC(C)=C(OC(=O)O)C1c1ccccc1OCc1c(Cl)cccc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 4/20 0.42
GAA P10253 4/20 0.42
CYP2C9 P11712 3/20 0.39
HSD17B10 Q99714 3/20 0.39
MEN1 O00255 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C19 P33261 2/20 0.39
KMT2A Q03164 2/20 0.39
HIF1A Q16665 2/20 0.39
NR1I2 O75469 2/20 0.39
ABCB11 O95342 2/20 0.39
MAPT P10636 2/20 0.39
HPGD P15428 2/20 0.39
TP53 P04637 1/20 0.39
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.39
NFKB1 P19838 1/20 0.39
THPO P40225 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10817440 0.94 ALDH1A1 (0.47) ALDH1A1KDM4EGAACYP2C9HSD17B10
SCHEMBL9691465 0.91 ALDH1A1 (0.44) ALDH1A1KDM4EGAACYP2C9HSD17B10
SCHEMBL9690847 0.90 FABP4 (0.45) KDM4EGAANR1I2TP53LMNA
SCHEMBL9691359 0.87 POLB (0.44) ALDH1A1KDM4EGAAHSD17B10MEN1
SCHEMBL10649148 0.86 HPGD (0.41) ALDH1A1KDM4EGAACYP2C9HSD17B10
SCHEMBL9690877 0.86 HTR6 (0.43) KDM4EGAANR1I2MAPTSLC6A3
SCHEMBL10374975 0.84 ALDH1A1 (0.46) ALDH1A1KDM4EGAACYP2C9HSD17B10
SCHEMBL9691648 0.84 TP53 (0.41) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL10914095 0.83 POLB (0.46) ALDH1A1KDM4EGAAHSD17B10MEN1
SCHEMBL9691625 0.83 NR1I2 (0.42) ALDH1A1KDM4EGAAKMT2ANR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0071819-B2 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1992-06-10 EP disclosed
EP-0288758-A2 Dihydropyridinamides, process for their preparation and their use in medicines BAYER AG (DE) 1988-11-02 EP disclosed