SCHEMBL9700197

SCHEMBL9700197

CC(C)=CCN1Cc2cccc([N+](=O)[O-])c2NCC1c1ccc(Cl)c(Cl)c1

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.32
SLC6A2 P23975 8/20 0.31
SLC6A4 P31645 8/20 0.31
SLC6A3 Q01959 5/20 0.31
CCR2 P41597 2/20 0.31
KDM4E B2RXH2 2/20 0.31
LMNA P02545 2/20 0.31
KMT2A Q03164 2/20 0.31
ALDH1A1 P00352 2/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
ALOX12 P18054 1/20 0.31
MAPK1 P28482 1/20 0.31
RECQL P46063 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
POLB P06746 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30
TAS1R3 Q7RTX0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9701430 0.90 CA1 (0.33) MAOBLMNANPC1GAAMAPT
SCHEMBL9701113 0.88 MAOB (0.31) MAOBABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9701174 0.84 SLC6A2 (0.36) SLC6A2SLC6A4SLC6A3
SCHEMBL9535908 0.81 CHRNB2 (0.34) KMT2AMAPK1L3MBTL1TAS1R3TAS1R1
SCHEMBL9436772 0.81 CHRNB2 (0.34) KMT2AMAPK1L3MBTL1TAS1R3TAS1R1
SCHEMBL9702143 0.79 MAOB (0.32) MAOBKDM4E
SCHEMBL9702535 0.72 MAPT (0.35) KDM4ELMNAALDH1A1GAAMAPT
SCHEMBL7902272 0.71 KDM4E (0.32) KDM4EALDH1A1POLB
SCHEMBL9701097 0.70 SIGMAR1 (0.34) MAOBSLC6A2SLC6A4SLC6A3LMNA
SCHEMBL9702241 0.69 RAB9A (0.33) KDM4ELMNAKMT2AALDH1A1TAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992013860-A1 NEW 4,5,6,7-TETRAHYDRO-IMIDAZO-[4,5,lJK][1,4]-BENZODIAZEPINE-2-(1H)-THIONES, A METHOD OF PREPARING THEM AS WELL AS DRUGS CONTAINING THEM, AND INTERMEDIATES FOR THE PREPARATION OF THESE COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1992-08-20 WO disclosed