SCHEMBL9702535

SCHEMBL9702535

COc1ccc(CC2CNc3c(cccc3[N+](=O)[O-])CN2CC=C(C)C)cc1OC

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.35
TAAR1 Q96RJ0 1/20 0.35
ALDH1A1 P00352 4/20 0.35
HCRTR1 O43613 3/20 0.34
HCRTR2 O43614 3/20 0.34
HTT P42858 2/20 0.34
GAA P10253 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPK1 P28482 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
TTR P02766 1/20 0.34
LMNA P02545 1/20 0.34
GALR3 O60755 1/20 0.34
NR2F2 P24468 1/20 0.34
RAB9A P51151 1/20 0.34
CYP19A1 P11511 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9535908 0.78 CHRNB2 (0.34) MAPK1L3MBTL1RAB9ACYP1A2CYP3A4
SCHEMBL9701397 0.77 CA1 (0.33) MAPTALDH1A1HCRTR1HCRTR2HTT
SCHEMBL9701430 0.73 CA1 (0.33) MAPTHTTGAALMNARAB9A
SCHEMBL9700197 0.72 MAOB (0.32) MAPTALDH1A1GAAKDM4EMAPK1
SCHEMBL9702700 0.70 SIGMAR1 (0.33) ALDH1A1
SCHEMBL9702241 0.67 RAB9A (0.33) ALDH1A1KDM4ELMNARAB9ACYP3A4
SCHEMBL7902260 0.65 CYP1A2 (0.35) MAPTALDH1A1KDM4EMAPK1L3MBTL1
SCHEMBL7902256 0.65 CYP1A2 (0.35) MAPTALDH1A1KDM4EMAPK1L3MBTL1
SCHEMBL9702570 0.65 MAPT (0.42) MAPTALDH1A1HTTKDM4EMAPK1
SCHEMBL9702143 0.62 MAOB (0.32) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992013860-A1 NEW 4,5,6,7-TETRAHYDRO-IMIDAZO-[4,5,lJK][1,4]-BENZODIAZEPINE-2-(1H)-THIONES, A METHOD OF PREPARING THEM AS WELL AS DRUGS CONTAINING THEM, AND INTERMEDIATES FOR THE PREPARATION OF THESE COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1992-08-20 WO disclosed