SCHEMBL9700327

SCHEMBL9700327

CNCC1COc2c(OC)cccc2N1N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 11/20 0.38
ADRA1A P35348 11/20 0.38
ADRA1B P35368 11/20 0.38
HTR1A P08908 3/20 0.34
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP2C19 P33261 1/20 0.34
THPO P40225 1/20 0.34
KMT2A Q03164 1/20 0.34
ADRA2A P08913 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10378979 0.87 ADRA1A (0.38) ADRA1DADRA1AADRA1BHTR1AALDH1A1
SCHEMBL9700158 0.85 HTR2A (0.38) ADRA1DADRA1AADRA1BHTR1AKDM4E
SCHEMBL9700368 0.82 NOTUM (0.37) ADRA1DADRA1AADRA1BCYP2D6SLC6A2
SCHEMBL9701394 0.81 ADRA1A (0.36) ADRA1DADRA1AADRA1BKDM4EADRA2A
SCHEMBL9700351 0.80 ADRA2A (0.41) ADRA1DADRA1AADRA1BHTR1AALDH1A1
SCHEMBL9701613 0.80 ADRA2A (0.41) ADRA1DADRA1AADRA1BHTR1AADRA2A
SCHEMBL10471313 0.79 ADRA2A (0.37) ADRA1DADRA1AADRA1BHTR1AALDH1A1
SCHEMBL9699337 0.78 ADRA2A (0.42) ADRA1DADRA1AADRA1BHTR1AADRA2A
SCHEMBL9728617 0.77 ADRA1A (0.41) ADRA1DADRA1AADRA1BHTR1AALDH1A1
SCHEMBL9699287 0.74 HTR7 (0.40) ADRA1DADRA1AADRA1BHTR1ACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed