SCHEMBL9701293

SCHEMBL9701293

CCCc1cc(-c2ccc(C#N)c(=O)[nH]2)cc(Br)c1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
KDM4E B2RXH2 4/20 0.50
GLA P06280 3/20 0.50
GAA P10253 2/20 0.50
L3MBTL1 Q9Y468 2/20 0.50
PDE3B Q13370 2/20 0.38
PDE3A Q14432 2/20 0.38
GPR35 Q9HC97 2/20 0.37
PIM1 P11309 1/20 0.37
MDM2 Q00987 1/20 0.36
HPGD P15428 2/20 0.36
CYP1A2 P05177 1/20 0.36
HSD17B10 Q99714 1/20 0.36
IDH1 O75874 4/20 0.34
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
KMT2A Q03164 1/20 0.33
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9526437 0.81 ALDH1A1 (0.45) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9701626 0.81 ALDH1A1 (0.56) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9700723 0.75
SCHEMBL9701665 0.75 KDM4E (0.61) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9701832 0.73 KDM4E (0.77) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9525396 0.72 ALDH1A1 (0.49) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9525387 0.72 ALDH1A1 (0.49) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9526579 0.72 KDM4E (0.56) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9526574 0.72 KDM4E (0.56) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9524981 0.71 KDM4E (0.54) ALDH1A1KDM4EGLAGAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992006085-A1 PHENYLPYRIDINOL DERIVATIVES AS MEDICAMENTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1992-04-16 WO disclosed