SCHEMBL9701626

SCHEMBL9701626

CCCc1cc(-c2ccc(C#N)c(=O)[nH]2)ccc1OC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.56
KDM4E B2RXH2 3/20 0.56
GLA P06280 2/20 0.56
GAA P10253 2/20 0.56
L3MBTL1 Q9Y468 2/20 0.56
GABRA1 P14867 2/20 0.42
GABRB2 P47870 2/20 0.42
ALOX5 P09917 1/20 0.42
PIM1 P11309 2/20 0.41
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
GABRA5 P31644 1/20 0.40
GABRA3 P34903 1/20 0.40
GABRA2 P47869 1/20 0.40
AR P10275 2/20 0.40
MAPK1 P28482 1/20 0.39
CHEK1 O14757 1/20 0.38
MDM2 Q00987 1/20 0.38
CYP1A2 P05177 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9701530 0.83 KDM4E (0.65) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9526844 0.82 KDM4E (0.55) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9701620 0.82 KDM4E (0.57) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9701293 0.81 ALDH1A1 (0.50) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9701665 0.80 KDM4E (0.61) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9701460 0.78 ALDH1A1 (0.52) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9701927 0.78 KDM4E (0.55) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL7371751 0.77 KDM4E (0.57) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL7371748 0.77 KDM4E (0.57) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9526258 0.77 KDM4E (0.64) ALDH1A1KDM4EGLAGAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992006085-A1 PHENYLPYRIDINOL DERIVATIVES AS MEDICAMENTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1992-04-16 WO disclosed