SCHEMBL9526437

SCHEMBL9526437

CCCc1cc(-c2ccc(C#N)c(=O)[nH]2)cc(NC(C)=O)c1OC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
KDM4E B2RXH2 2/20 0.45
GLA P06280 1/20 0.45
GAA P10253 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
GABRA1 P14867 2/20 0.41
GABRB2 P47870 2/20 0.41
PDE3B Q13370 2/20 0.35
PDE3A Q14432 2/20 0.35
MET P08581 1/20 0.34
KDR P35968 1/20 0.34
MDM2 Q00987 1/20 0.33
STK4 Q13043 1/20 0.33
PDE5A O76074 1/20 0.32
PDE4A P27815 1/20 0.32
PDE1A P54750 1/20 0.32
PDE1B Q01064 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9701293 0.81 ALDH1A1 (0.50) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9525349 0.78 ALDH1A1 (0.44) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9526870 0.78 GABRA1 (0.40) GABRA1GABRB2PDE3BPDE3APDE5A
SCHEMBL9701626 0.76 ALDH1A1 (0.56) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL11118460 0.70 PGR (0.49) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL11110995 0.69 ALDH1A1 (0.58) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9701832 0.68 KDM4E (0.77) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9525396 0.68 ALDH1A1 (0.49) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9525387 0.68 ALDH1A1 (0.49) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL9526574 0.67 KDM4E (0.56) ALDH1A1KDM4EGLAGAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0550576-A1 PHENYLPYRIDINOL DERIVATIVES AS MEDICAMENTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1993-07-14 EP disclosed
WO-1992006085-A1 PHENYLPYRIDINOL DERIVATIVES AS MEDICAMENTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1992-04-16 WO disclosed