SCHEMBL9701625

SCHEMBL9701625

C=C=C(CN)Cc1cccc(O)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.55
DRD1 P21728 2/20 0.55
TAAR1 Q96RJ0 1/20 0.55
ENPP2 Q13822 1/20 0.53
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
PKM P14618 1/20 0.44
ALOX15 P16050 1/20 0.44
NFKB1 P19838 1/20 0.44
MAPK1 P28482 1/20 0.44
KMT2A Q03164 1/20 0.43
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
CTBP2 P56545 1/20 0.41
MIF P14174 1/20 0.39
DRD4 P21917 1/20 0.39
DRD5 P21918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10442128 0.82 ACHE (0.38) DRD2DRD1TAAR1ENPP2CYP3A4
SCHEMBL9701924 0.80 LOXL2 (0.43) TAAR1
Hydrochloric Acid SCHEMBL11493475 0.78 LOXL2 (0.41) TAAR1
SCHEMBL9702029 0.78 TAAR1 (0.48) TAAR1KMT2AKDM4EBLM
SCHEMBL9701928 0.77 KDM4E (0.53) DRD2DRD1TAAR1CYP1A2CYP3A4
SCHEMBL9701911 0.73 TAAR1 (0.35) TAAR1ALOX15KDM4ELMNAMAPT
SCHEMBL9702218 0.72 APP (0.43) DRD2DRD1TAAR1ENPP2MAPK1
SCHEMBL43719 0.71 TAAR1 (1.00) DRD2DRD1TAAR1ENPP2CYP1A2
SCHEMBL29465557 0.71 TAAR1 (1.00) DRD2DRD1TAAR1ENPP2CYP1A2
SCHEMBL29598265 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5120764-A Administering penicillamine and allenylamines to inhibit crosslinking of collagen MERRELL DOW PHARMACEUTICALS INC. (US) 1992-06-09 US disclosed
EP-0374440-A2 Inhibitors of lysyl oxidase MERRELL DOW PHARMACEUTICALS INC. (US) 1990-06-27 EP disclosed