SCHEMBL9701802

SCHEMBL9701802

NC(=O)N(O)CCn1cc(Cc2ccccc2)c2ccccc21

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 7/20 0.64
HDAC3 O15379 1/20 0.55
HDAC1 Q13547 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
ICMT O60725 1/20 0.44
KRAS P01116 1/20 0.43
CDC25A P30304 1/20 0.43
KMT2A Q03164 1/20 0.41
ALDH1A1 P00352 2/20 0.40
CREBBP Q92793 1/20 0.40
POLB P06746 1/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7808063 0.88 HTR6 (0.50) HTR6HDAC3HDAC1HDAC8HDAC6
SCHEMBL7809786 0.80 HDAC3 (0.50) HTR6HDAC3ICMTCDC25ALMNA
SCHEMBL3328890 0.79 HTR6 (1.00) HTR6HDAC3
SCHEMBL9701525 0.77 ALDH1A1 (0.44) KMT2AALDH1A1CREBBPPOLBSMN1; SMN2
SCHEMBL9701519 0.76 KMT2A (0.60) HTR6HDAC3HDAC1HDAC8HDAC6
SCHEMBL7815554 0.74 HDAC1 (0.49) HTR6HDAC3HDAC1HDAC8HDAC6
SCHEMBL12850648 0.73 HDAC6 (0.74) HDAC3HDAC1HDAC8HDAC6KMT2A
SCHEMBL9701366 0.73 HTR6 (0.62) HTR6HDAC3HDAC1HDAC8HDAC6
SCHEMBL28313770 0.72 HDAC1 (0.68) HTR6HDAC1HDAC8HDAC6KMT2A
SCHEMBL7811888 0.71 CAMK2D (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132319-A Antiasthmatic, antiinflammatory, antiallergen and cytoprotective agents MERCK FROSST CANADA, INC. (CA) 1992-07-21 US disclosed