SCHEMBL11021898

SCHEMBL11021898

COc1cc(S(C)(=O)=O)ccc1-c1nc2ccc(C#N)cc2[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.53
CDK4 P11802 1/20 0.49
CCNA2 P20248 1/20 0.49
CCND1 P24385 1/20 0.49
CDK2 P24941 1/20 0.49
CCND3 P30281 1/20 0.49
NPBWR1 P48145 1/20 0.48
SCD O00767 5/20 0.46
PKN1 Q16512 1/20 0.46
PKN2 Q16513 1/20 0.46
CBFB Q13951 1/20 0.45
CFB P00751 3/20 0.44
FADS1 O60427 1/20 0.44
CHEK2 O96017 1/20 0.44
METAP2 P50579 1/20 0.44
METAP1 P53582 1/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11021893 0.91 ATR (0.44) ATRCDK4CCNA2CCND1CDK2
SCHEMBL11020318 0.90 CA12 (0.54) ATRSCDPKN1PKN2CFB
SCHEMBL11018186 0.89 CYP3A4 (0.48) ATRSCDPKN1PKN2CFB
SCHEMBL11016115 0.89 CFB (0.47) ATRPKN1PKN2CFBCHEK2
SCHEMBL11022217 0.89 ATR (0.53) ATRNPBWR1SCDPKN1PKN2
SCHEMBL11018866 0.89 MAPT (0.44) ATRCDK4CCNA2CCND1CDK2
SCHEMBL11018077 0.87 CYP2C9 (0.54) ATRPKN1PKN2CFBCHEK2
SCHEMBL11021561 0.84 L3MBTL1 (0.47) ATRPKN1PKN2CFBCHEK2
SCHEMBL11017639 0.84 MAPT (0.49) ATRPKN1PKN2CFB
SCHEMBL10580157 0.84 CDK4 (0.47) CDK4CCNA2CCND1CDK2CCND3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0148431-A1 Benzimidazoles, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-07-17 EP claimed
EP-0148431-A1 Benzimidazoles, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-07-17 EP disclosed