SCHEMBL9702964

SCHEMBL9702964

Nc1cccc(O)c1-c1ccc2cc(I)ccc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 6/20 0.40
HSD17B2 P37059 6/20 0.40
CYP3A4 P08684 5/20 0.40
CYP1A2 P05177 4/20 0.40
CYP2D6 P10635 4/20 0.40
CYP2C9 P11712 4/20 0.40
CYP2B6 P20813 4/20 0.40
CYP2C19 P33261 4/20 0.40
ESR2 Q92731 8/20 0.37
ESR1 P03372 7/20 0.36
ALOX5 P09917 1/20 0.36
ALOX15 P16050 3/20 0.35
TSHR P16473 1/20 0.35
CTDSP1 Q9GZU7 1/20 0.35
HSD17B10 Q99714 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2934548 0.85 ALOX5 (0.52) HSD17B1HSD17B2CYP3A4CYP1A2CYP2D6
SCHEMBL9702969 0.77 ESR2 (0.47) HSD17B1HSD17B2CYP3A4CYP1A2CYP2D6
SCHEMBL2937944 0.75 APP (0.54) HSD17B1HSD17B2CYP3A4CYP1A2CYP2D6
SCHEMBL2937981 0.75 ALDH1A1 (0.57) HSD17B1HSD17B2CYP3A4CYP1A2CYP2D6
SCHEMBL2938310 0.75 MEN1 (0.50) HSD17B1HSD17B2CYP3A4CYP1A2CYP2D6
SCHEMBL9319110 0.73 CYP1A2 (0.52) HSD17B1HSD17B2CYP3A4CYP1A2ESR2
SCHEMBL2937291 0.72 HSD17B1 (0.50) HSD17B1HSD17B2CYP3A4CYP1A2CYP2D6
SCHEMBL2931315 0.72 CYP3A4 (0.50) HSD17B1HSD17B2CYP3A4CYP1A2CYP2D6
SCHEMBL2937049 0.71 MCL1 (0.41) HSD17B1HSD17B2CYP3A4ESR2ALOX15
SCHEMBL2935347 0.71 ALOX15 (0.46) CYP3A4ALOX15TSHRCTDSP1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0221677-B1 P-AMINOPHENOLS, DERIVATIVES THEREOF AND USE FOR MANUFACTURE OF A MEDICAMENT E.R. Squibb & Sons, Inc. (US) 1992-09-09 EP claimed
US-4910208-A Skin disorders, antiinflammatory agent E. R. SQUIBB & SONS, INC. (US) 1990-03-20 US claimed
EP-0221677-A2 p-Aminophenols, derivatives thereof and use for manufacture of a medicament E.R. Squibb & Sons, Inc. (US) 1987-05-13 EP claimed