SCHEMBL9702969

SCHEMBL9702969

Nc1c(O)cccc1-c1ccc2cc(I)ccc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 8/20 0.47
HDAC4 P56524 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
ESR1 P03372 7/20 0.36
HSD17B1 P14061 5/20 0.36
HSD17B2 P37059 5/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2B6 P20813 1/20 0.36
ALOX5 P09917 1/20 0.36
APP P05067 1/20 0.35
CTDSP1 Q9GZU7 1/20 0.35
GSTP1 P09211 1/20 0.33
DHFR P00374 1/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28618814 0.85 ESR2 (0.56) ESR2HDAC4HDAC2HDAC8ESR1
SCHEMBL9702964 0.77 HSD17B1 (0.40) ESR2ESR1HSD17B1HSD17B2CYP1A2
SCHEMBL27877792 0.72 HSD17B1 (0.50) ESR2ESR1HSD17B1HSD17B2CYP1A2
SCHEMBL3790386 0.72 MAP4K4 (0.50) HSD17B1HSD17B2CYP1A2CYP2C9CYP2C19
SCHEMBL30439996 0.72 HSD17B1 (0.50) ESR2ESR1HSD17B1HSD17B2CYP1A2
SCHEMBL13670758 0.71 MCL1 (0.46) ESR2HDAC4HDAC2HDAC8CYP1A2
SCHEMBL3789766 0.71 ALDH1A1 (0.43) CYP3A4APPCTDSP1MEN1LMNA
SCHEMBL19880343 0.70 ESR1 (0.44) ESR2ESR1HSD17B1HSD17B2CYP1A2
SCHEMBL564030 0.70 CASP7 (0.50) CYP1A2CYP3A4CTDSP1MEN1LMNA
SCHEMBL565555 0.69 ALDH1A1 (0.62) HDAC4HDAC2HDAC8HSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0221677-B1 P-AMINOPHENOLS, DERIVATIVES THEREOF AND USE FOR MANUFACTURE OF A MEDICAMENT E.R. Squibb & Sons, Inc. (US) 1992-09-09 EP claimed
US-4910208-A Skin disorders, antiinflammatory agent E. R. SQUIBB & SONS, INC. (US) 1990-03-20 US claimed
EP-0221677-A2 p-Aminophenols, derivatives thereof and use for manufacture of a medicament E.R. Squibb & Sons, Inc. (US) 1987-05-13 EP claimed