SCHEMBL9707712

SCHEMBL9707712

COC(C)n1c(=O)[nH]c(=O)c2c1nc(C(C)C)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.40
ALDH1A1 P00352 4/20 0.40
HPGD P15428 2/20 0.40
MAPT P10636 2/20 0.40
GAA P10253 1/20 0.40
HTT P42858 1/20 0.40
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
NPSR1 Q6W5P4 2/20 0.37
CXCL8 P10145 1/20 0.36
NOD2 Q9HC29 1/20 0.36
NOD1 Q9Y239 1/20 0.36
USP1 O94782 4/20 0.36
PPARG P37231 1/20 0.35
PKM P14618 2/20 0.35
MCL1 Q07820 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707480 0.91 KDM4E (0.42) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL9707838 0.90 AGTR1 (0.43) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL9707862 0.89 PPARG (0.37) USP1PPARG
SCHEMBL9708293 0.89 USP1 (0.39) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL9707565 0.88 AGTR1 (0.44) MEN1KMT2APPARG
SCHEMBL9708044 0.88 ALDH1A1 (0.38) ALDH1A1HPGDMAPTUSP1HSD17B10
SCHEMBL9708637 0.88 PPARG (0.37) USP1PPARG
SCHEMBL9708625 0.88 ALDH1A1 (0.38) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL9708130 0.88 CXCL8 (0.49) KDM4EALDH1A1HPGDMAPTHTT
SCHEMBL9707740 0.87 PPARG (0.35) PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed