SCHEMBL9707971

SCHEMBL9707971

C=C(CC)c1nc2c(c(=O)n(C)c(=O)n2CCC)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.38
ADORA3 P0DMS8 4/20 0.37
AGTR1 P30556 2/20 0.36
AGTR2 P50052 1/20 0.36
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
GPR18 Q14330 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707888 0.95 ADORA3 (0.41) ADORA3ADORA2AADORA1
SCHEMBL9707710 0.92 MAPT (0.39) HPGDLMNASMN1; SMN2
SCHEMBL9708256 0.88 HPGD (0.44) HPGDADORA3ADORA2A
SCHEMBL9707666 0.88 ADORA3 (0.42) ADORA3ADORA2AADORA1
SCHEMBL9707689 0.88 TRPC5 (0.45) ADORA3
SCHEMBL9707817 0.86 AGTR1 (0.44) HPGDAGTR1AGTR2LMNA
SCHEMBL9707374 0.85 AGTR1 (0.46) AGTR1AGTR2
SCHEMBL9707814 0.85 ADORA3 (0.42) HPGDADORA3AGTR1AGTR2LMNA
SCHEMBL9707771 0.84 ALDH1A1 (0.45) AGTR1AGTR2LMNASMN1; SMN2
SCHEMBL9707907 0.84 GPR18 (0.37) HPGDAGTR1AGTR2GPR18

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO claimed
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed