SCHEMBL9708256

SCHEMBL9708256

CCCn1c(=O)n(C)c(=O)c2c1nc(C)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.44
ADORA2B P29275 3/20 0.41
ADORA2A P29274 1/20 0.41
ADORA3 P0DMS8 7/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707525 0.95 ADORA2B (0.46) ADORA2BADORA2AADORA3
SCHEMBL9708690 0.93 MAPT (0.42) ADORA2BADORA2AADORA3
SCHEMBL9708836 0.91 HPGD (0.47) HPGD
SCHEMBL9708711 0.91 ALOX15 (0.46)
SCHEMBL9708117 0.91 DCTPP1 (0.43) HPGDADORA3
SCHEMBL9707817 0.90 AGTR1 (0.44) HPGD
SCHEMBL9707423 0.90 ADORA3 (0.42) ADORA2BADORA2AADORA3
SCHEMBL9708509 0.90 ADORA3 (0.40) ADORA2BADORA2AADORA3
SCHEMBL9708336 0.90 ADORA3 (0.46) ADORA2BADORA2AADORA3
SCHEMBL9707551 0.90 ADORA3 (0.46) ADORA2BADORA2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed