SCHEMBL9708313

SCHEMBL9708313

COC(=O)Cn1c(=O)[nH]c(=O)c2c1nc(CC(C)(C)C)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.44
KMT2A Q03164 5/20 0.44
NPSR1 Q6W5P4 2/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
TPH2 Q8IWU9 8/20 0.44
TPH1 P17752 7/20 0.44
AGTR1 P30556 1/20 0.41
AGTR2 P50052 1/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
POLB P06746 1/20 0.38
PPARG P37231 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708525 0.92 TPH2 (0.47) MEN1KMT2ANPSR1CYP3A4CYP2C9
SCHEMBL9708175 0.90 AGTR1 (0.48) MEN1KMT2ANPSR1CYP3A4CYP2C9
SCHEMBL9707753 0.89 AGTR1 (0.43) KMT2AAGTR1AGTR2PPARG
SCHEMBL9707900 0.89 AGTR1 (0.43) MEN1KMT2ACYP2C9CYP2C19AGTR1
SCHEMBL9707269 0.89 MEN1 (0.51) MEN1KMT2ATPH2TPH1
SCHEMBL9708417 0.89 AGTR2 (0.53) MEN1KMT2AAGTR1AGTR2PPARG
SCHEMBL9708631 0.89 ALDH1A1 (0.47) MEN1KMT2ANPSR1TPH2TPH1
SCHEMBL9707246 0.88 MEN1 (0.46) MEN1KMT2ANPSR1CYP3A4CYP2C9
SCHEMBL9708139 0.88 TSHR (0.42) MEN1KMT2ANPSR1CYP2C9CYP2C19
SCHEMBL9708081 0.88 AGTR1 (0.51) MEN1KMT2ANPSR1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed