SCHEMBL9713868

SCHEMBL9713868

N#Cc1cc(S(=O)(=O)c2ccc(N)cc2)ccc1N

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.62
ALDH1A1 P00352 4/20 0.62
PKM P14618 2/20 0.62
LMNA P02545 3/20 0.55
TSHR P16473 3/20 0.55
CYP3A4 P08684 2/20 0.55
CYP2C9 P11712 2/20 0.55
MPO P05164 1/20 0.55
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
NPC1 O15118 1/20 0.44
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
CYP2C19 P33261 2/20 0.40
KDM4E B2RXH2 2/20 0.40
CYP2D6 P10635 1/20 0.40
CA12 O43570 1/20 0.39
USP2 O75604 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL591137 0.88 ALDH1A1 (0.51) HTR6ALDH1A1PKMLMNATSHR
SCHEMBL1700011 0.80 CA2 (0.55) ALDH1A1PKMLMNATSHRCYP2C9
SCHEMBL7991225 0.79 ALDH1A1 (0.52) ALDH1A1PKMLMNATSHRCYP3A4
SCHEMBL2577731 0.79 G6PD (0.53) TSHRCYP3A4CYP2C9CYP2C19KDM4E
SCHEMBL30771551 0.77 HTR6 (1.00) HTR6ALDH1A1PKMLMNATSHR
SCHEMBL728291 0.77 HTR6 (1.00) HTR6ALDH1A1PKMLMNATSHR
SCHEMBL9713772 0.76 HTR6 (0.50) HTR6ALDH1A1PKMLMNATSHR
SCHEMBL20379869 0.76 HTR6 (0.67) HTR6ALDH1A1PKMLMNATSHR
Dapsone SCHEMBL2590728 0.75 HTR6 (0.73) HTR6ALDH1A1PKMLMNATSHR
SCHEMBL15393731 0.75 POLB (0.42) HTR6ALDH1A1PKMTSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084449-A Bactericides and antiprotozoa agents DR. KARL THOMAE GMBH (DE) 1992-01-28 US disclosed
US-4992430-A Anti-bacterial compositions comprising a substituted bis-(4-aminophenyl)-sulfone and a dihydro-folic acid reductase DR. KARL THOMAE GMBH (DE) 1991-02-12 US disclosed
US-4829058-A INHIBITORS OF BACTERIA, MYCOBACTERIA AND PLASMODIA DR. KARL THOMAE GMBH (DE) 1989-05-09 US disclosed
EP-0165422-B1 SUBSTITUTED BIS-(4-AMINOPHENYL)-SULPHONES, THEIR PREPARATION AND THEIR USE AS MEDICINES Dr. Karl Thomae GmbH (DE) 1988-03-09 EP disclosed
EP-0165422-A1 Substituted bis-(4-aminophenyl)-sulphones, their preparation and their use as medicines Dr. Karl Thomae GmbH (DE) 1985-12-27 EP disclosed