SCHEMBL9720646

SCHEMBL9720646

COc1ccccc1C(c1ccccc1OC)N1CCN(Cc2ccc(O)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
TSHR P16473 1/20 0.53
CYP2C19 P33261 1/20 0.53
KMT2A Q03164 2/20 0.51
MAPK1 P28482 1/20 0.49
OPRM1 P35372 1/20 0.49
OPRD1 P41143 1/20 0.49
OPRK1 P41145 1/20 0.49
OPRL1 P41146 1/20 0.49
KDM4E B2RXH2 1/20 0.48
SIGMAR1 Q99720 1/20 0.48
ATM Q13315 2/20 0.47
MEN1 O00255 1/20 0.47
DRD4 P21917 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9720740 0.84 ATM (0.48) CYP1A2CYP3A4CYP2D6CYP2C19KMT2A
SCHEMBL9720772 0.82 OPRM1 (0.50) KMT2AOPRM1OPRD1OPRK1OPRL1
SCHEMBL9720688 0.81 OPRD1 (0.50) ALDH1A1KMT2AOPRD1OPRK1KDM4E
SCHEMBL9720681 0.78 MAPK1 (0.78) ALDH1A1KMT2AMAPK1KDM4EDRD4
Belarizine SCHEMBL2108057 0.77 ATM (0.73) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL9720800 0.77 SIGMAR1 (0.56) KMT2AMAPK1OPRD1OPRK1SIGMAR1
SCHEMBL9720680 0.76 SIGMAR1 (0.54) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL25861444 0.74 HRH3 (0.56) ALDH1A1KMT2AKDM4EMEN1DRD4
SCHEMBL9720718 0.73 TRPV6 (0.58) ALDH1A1KMT2AKDM4EATMMEN1
SCHEMBL9720752 0.73 DRD4 (0.77) KMT2ASIGMAR1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5142052-A Cationic effect-driven carbinol/amine reaction LABORATOIRES SYNTEX (FR) 1992-08-25 US disclosed