SCHEMBL9727649

SCHEMBL9727649

c1ccc(CCC2Cc3cc(OCc4ccccc4)c(CCCOc4ccc(-c5nnn[nH]5)cc4)cc3O2)cc1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.34
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
ABCB1 P08183 1/20 0.33
HTR6 P50406 1/20 0.32
BRD4 O60885 1/20 0.32
CREBBP Q92793 1/20 0.32
PRMT5 O14744 1/20 0.32
GP6 Q9HCN6 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727749 0.89 MAOA (0.34) MAOAMAOBBRD4CREBBPGP6
SCHEMBL5502488 0.85 MAOA (0.40) MAOAMAOBHTR6
SCHEMBL9727339 0.81 MAOB (0.43) MAOAMAOBHTR6
SCHEMBL9727458 0.81 PTGER1 (0.47)
SCHEMBL5513024 0.79 HPGD (0.32)
SCHEMBL9727691 0.79 MTNR1B (0.42)
SCHEMBL9727567 0.77 CYP3A4 (0.37) HTR6
SCHEMBL14435033 0.77 HTR6 (0.43) HTR6
SCHEMBL9727767 0.76 HIF1A (0.36) HIF1A
SCHEMBL9727765 0.76 MTNR1B (0.39) HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed