SCHEMBL9727339

SCHEMBL9727339

N#Cc1ccc(OCCCc2cc3c(cc2OCc2ccccc2)CC(CCc2ccccc2)O3)cc1

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.43
MAOA P21397 3/20 0.38
HTR6 P50406 1/20 0.35
AR P10275 1/20 0.34
MET P08581 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5502488 0.92 MAOA (0.40) MAOBMAOAHTR6
SCHEMBL9727458 0.87 PTGER1 (0.47)
SCHEMBL9727691 0.84 MTNR1B (0.42)
SCHEMBL9727567 0.83 CYP3A4 (0.37) HTR6
SCHEMBL14435033 0.83 HTR6 (0.43) HTR6
SCHEMBL9727649 0.81 HIF1A (0.34) MAOBMAOAHTR6
SCHEMBL9727765 0.81 MTNR1B (0.39)
SCHEMBL9727767 0.81 HIF1A (0.36)
SCHEMBL5518490 0.80 F2 (0.41) MAOBMAOA
SCHEMBL9727664 0.80 MAPK1 (0.38) MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed