SCHEMBL9727664

SCHEMBL9727664

O=C(COc1cc2c(cc1CCCOc1ccccc1)OC(CCc1ccccc1)C2)OCc1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CASP1 P29466 1/20 0.37
KDM4E B2RXH2 2/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
HPGD P15428 1/20 0.34
ATM Q13315 1/20 0.34
HSD17B10 Q99714 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5518490 0.90 F2 (0.41) MAOAMAOBMTNR1AMTNR1B
SCHEMBL9727458 0.86 PTGER1 (0.47)
SCHEMBL9727691 0.83 MTNR1B (0.42) NPC1RAB9ASMN1; SMN2MTNR1B
SCHEMBL14435032 0.81 MTNR1A (0.38) MTNR1AMTNR1B
SCHEMBL9727339 0.80 MAOB (0.43) MAOAMAOB
SCHEMBL5506271 0.80 MAOA (0.41) MAOAMAOB
SCHEMBL14435047 0.80 F2 (0.39) MAPK1NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL9727767 0.80 HIF1A (0.36) NPC1RAB9ASMN1; SMN2MTNR1AMTNR1B
SCHEMBL14435033 0.79 HTR6 (0.43)
SCHEMBL9727567 0.77 CYP3A4 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed