SCHEMBL9727705

SCHEMBL9727705

C=CCc1cc2c(cc1OCc1ccccc1)C(C)C(Cc1ccc(OC)cc1)O2

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.41
BCHE P06276 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
CYP3A4 P08684 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
ALOX12 P18054 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
SIRT2 Q8IXJ6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727488 0.84 ABCB1 (0.43) ABCB1HTR1ADRD2
SCHEMBL9727672 0.84 ABCB1 (0.43) ABCB1HTR1ADRD2
SCHEMBL9727708 0.81 ALDH1A1 (0.42) ALDH1A1TP53CYP3A4ALOX15TSHR
SCHEMBL9727783 0.74 ALDH1A1 (0.42) MEN1KMT2AALDH1A1TP53CYP3A4
SCHEMBL21363609 0.74 CYP3A4 (0.48) BCHEALDH1A1TP53CYP3A4ALOX15
SCHEMBL4231254 0.73 MAOB (0.51) ABCB1BCHEMEN1KMT2AALDH1A1
SCHEMBL9727762 0.70 NR3C1 (0.38) ABCB1BCHEMEN1KMT2AALDH1A1
SCHEMBL9727495 0.69 ALDH1A1 (0.43) MEN1KMT2AALDH1A1CYP3A4SMN1; SMN2
SCHEMBL14552348 0.69 MAOB (0.54) MEN1KMT2AALDH1A1TP53CYP3A4
SCHEMBL27859426 0.67 ALOX5 (0.50) BCHEMEN1KMT2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed