SCHEMBL9727672

SCHEMBL9727672

COc1ccc(CC2Oc3cc(CCCOc4ccccc4)c(OCc4ccccc4)cc3C2C)cc1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.43
MTNR1A P48039 4/20 0.40
MTNR1B P49286 3/20 0.40
HTR1A P08908 1/20 0.39
DRD2 P14416 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727488 0.91 ABCB1 (0.43) ABCB1MTNR1AMTNR1BHTR1ADRD2
SCHEMBL9727632 0.86 DRD2 (0.39) DRD2
SCHEMBL9727705 0.84 ABCB1 (0.41) ABCB1HTR1ADRD2
SCHEMBL9727653 0.72 ABCB1 (0.38) ABCB1MTNR1AMTNR1BHTR1ADRD2
SCHEMBL9727737 0.69 ESR1 (0.42)
SCHEMBL9727331 0.69 MTNR1A (0.37) ABCB1MTNR1AMTNR1BHTR1ADRD2
SCHEMBL9727495 0.68 ALDH1A1 (0.43)
SCHEMBL5502488 0.67 MAOA (0.40) HTR1A
SCHEMBL9727464 0.66 KDM4E (0.36)
SCHEMBL553770 0.64 APP (0.69) ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed