SCHEMBL9727743

SCHEMBL9727743

OCCCc1cc2c(cc1OCc1ccccc1)CC(CCc1ccc(Cl)cc1)O2

nearest known ligand 0.62

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.40
LTA4H P09960 1/20 0.40
EPHX2 P34913 1/20 0.40
PTGER1 P34995 1/20 0.37
PTGER4 P35408 1/20 0.37
PTGER3 P43115 1/20 0.37
PTGER2 P43116 1/20 0.37
CCR5 P51681 1/20 0.36
DRD4 P21917 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14435033 0.94 HTR6 (0.43) HTR6LTA4HEPHX2PTGER1PTGER4
SCHEMBL9727620 0.91 CCR5 (0.38) PTGER1PTGER4PTGER3PTGER2CCR5
SCHEMBL9727567 0.84 CYP3A4 (0.37) HTR6PTGER1PTGER4PTGER3PTGER2
SCHEMBL14446494 0.83 HTR6 (0.38) HTR6CYP3A4
SCHEMBL14435032 0.83 MTNR1A (0.38) CYP3A4
SCHEMBL5502488 0.83 MAOA (0.40) HTR6CYP3A4
SCHEMBL9727764 0.81 IGF1R (0.35)
SCHEMBL9727728 0.80 NR1I2 (0.32)
SCHEMBL9727458 0.80 PTGER1 (0.47) PTGER1PTGER4PTGER3PTGER2
SCHEMBL14435039 0.78 AKR1B1 (0.40) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed