SCHEMBL9727728

SCHEMBL9727728

CC(C)(C)[Si](C)(C)Oc1cc2c(cc1CCCO)OC(CCc1ccc(Cl)cc1)C2

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.32
MAOA P21397 1/20 0.32
PTGS2 P35354 1/20 0.32
OPRK1 P41145 1/20 0.32
SLC6A3 Q01959 1/20 0.32
TP53 P04637 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
TBXA2R P21731 1/20 0.31
HRH4 Q9H3N8 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727516 0.85 NR1I2 (0.33) NR1I2MAOAPTGS2OPRK1SLC6A3
SCHEMBL9727743 0.80 HTR6 (0.40)
SCHEMBL9727764 0.80 IGF1R (0.35) TBXA2RHRH4HRH3
SCHEMBL14435033 0.73 HTR6 (0.43)
SCHEMBL14446494 0.73 HTR6 (0.38)
SCHEMBL9727620 0.73 CCR5 (0.38)
SCHEMBL14435032 0.71 MTNR1A (0.38)
SCHEMBL14435039 0.69 AKR1B1 (0.40)
SCHEMBL9727677 0.69 PTGDR2 (0.38) MAOA
SCHEMBL9727775 0.68 TBXA2R (0.45) SLC6A3TBXA2RHRH4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed