SCHEMBL9730191

SCHEMBL9730191

Cc1[nH]cnc1CN(C)C(=O)c1cn2c3c(cccc13)SCC2

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 3/20 0.37
HTR3E A5X5Y0 2/20 0.37
HTR3B O95264 2/20 0.37
HTR3D Q70Z44 2/20 0.37
HTR3C Q8WXA8 2/20 0.37
MCL1 Q07820 4/20 0.36
BCL2 P10415 3/20 0.32
GABRR1 P24046 1/20 0.32
PARP1 P09874 1/20 0.31
OPRD1 P41143 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
ADRA2C P18825 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
ADRA1A P35348 1/20 0.31
HTR2B P41595 1/20 0.31
KCNH2 Q12809 1/20 0.31
CASP6 P55212 1/20 0.31
CD44 P16070 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9681702 0.82 MTNR1A (0.41) HTR3AHTR3EHTR3BHTR3DHTR3C
Cadaverine Tartrate SCHEMBL7429503 0.77 MTNR1A (0.37) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL8962729 0.76 HTR3A (0.46) HTR3AHTR3EHTR3BHTR3DHTR3C
Hydrochloric Acid SCHEMBL9730401 0.73 HTR3A (0.38) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL7267047 0.73 HTR3A (0.66) HTR3AHTR3EHTR3BHTR3DHTR3C
Fumaric Acid SCHEMBL7273886 0.72 HTR3E (0.42) HTR3AHTR3EHTR3BHTR3DHTR3C
Maleic Acid SCHEMBL7273875 0.72 HTR3E (0.42) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL19779451 0.70 MCL1 (0.45) MCL1BCL2PARP1
SCHEMBL25600150 0.70 MCL1 (0.52) MCL1BCL2PARP1
SCHEMBL6325566 0.67 MCL1 (0.43) MCL1BCL2PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5102901-A 5-hydroxytrypamine receptor antaonists DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1992-04-07 US disclosed