SCHEMBL9681702

SCHEMBL9681702

Cc1[nH]cnc1CN(C)C(=O)c1cn2c3c(cccc13)CCC2

nearest known ligand 0.70

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 7/20 0.41
MTNR1B P49286 7/20 0.41
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR3E A5X5Y0 1/20 0.37
HTR3B O95264 1/20 0.37
HTR3A P46098 1/20 0.37
HTR3D Q70Z44 1/20 0.37
HTR3C Q8WXA8 1/20 0.37
OPA1 O60313 1/20 0.37
EIF5B O60841 1/20 0.37
MET P08581 1/20 0.37
HMOX2 P30519 1/20 0.37
CD44 P16070 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cadaverine Tartrate SCHEMBL7429503 0.94 MTNR1A (0.37) MTNR1AMTNR1BHTR2AHTR2CHTR3E
SCHEMBL7299112 0.83 HTR3E (0.57) MTNR1AMTNR1BHTR2AHTR2CHTR3E
SCHEMBL9730191 0.82 HTR3A (0.37) HTR2AHTR2CHTR3EHTR3BHTR3A
SCHEMBL7332932 0.82 MTNR1A (0.46) MTNR1AMTNR1BHTR2AHTR2CHTR3E
Hydrochloric Acid SCHEMBL9730401 0.81 HTR3A (0.38) HTR2AHTR2CHTR3EHTR3BHTR3A
Hydrochloric Acid SCHEMBL9729932 0.80 MCL1 (0.41) HTR2AHTR2CCD44
Fumaric Acid SCHEMBL7298751 0.78 HTR3E (0.52) MTNR1AMTNR1BHTR2AHTR2CHTR3E
Maleic Acid SCHEMBL7298744 0.78 HTR3E (0.52) MTNR1AMTNR1BHTR2AHTR2CHTR3E
SCHEMBL8962729 0.77 HTR3A (0.46) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7301618 0.75 MTNR1A (0.40) MTNR1AMTNR1BHTR2AHTR2COPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5114950-A Psychological disorders, anxiety, nausea and vomiting GLAXO GROUP LIMITED (GB) 1992-05-19 US claimed
JP-3128376-A None JP disclosed
US-5114950-A Psychological disorders, anxiety, nausea and vomiting GLAXO GROUP LIMITED (GB) 1992-05-19 US disclosed
JP-H03128376-A AMIDE DERIVATIVE GLAXO GROUP LTD 1991-05-31 JP disclosed