SCHEMBL9735648

SCHEMBL9735648

Fc1c(F)c(F)c(P(=Cc2ccccc2)(c2ccccc2)c2ccccc2)c(F)c1F

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 4/20 0.34
HSP90AA1 P07900 1/20 0.31
ALDH1A1 P00352 2/20 0.30
TSHR P16473 1/20 0.30
MAOB P27338 1/20 0.30
CYP2A6 P11509 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1132385 0.80 ALDH1A1 (0.39) NFE2L2HSP90AA1ALDH1A1TSHRMAOB
SCHEMBL9541494 0.75 NFE2L2 (0.52) NFE2L2ALDH1A1TSHR
SCHEMBL9735643 0.72 HSP90AA1 (0.33) NFE2L2HSP90AA1TSHR
Benzaldehyde SCHEMBL6051056 0.71 ALDH1A1 (0.61) HSP90AA1ALDH1A1TSHRMAOBCYP2A6
SCHEMBL9539397 0.68 ALDH1A1 (0.41) HSP90AA1ALDH1A1
SCHEMBL7200192 0.67 ESR1 (0.44) TSHR
SCHEMBL24193844 0.67 ESR1 (0.50) NFE2L2HSP90AA1ALDH1A1
SCHEMBL9538596 0.67 LMNA (0.42) NFE2L2ALDH1A1TSHRCYP2A6
SCHEMBL14269409 0.67 ALDH1A1 (0.42) HSP90AA1ALDH1A1MAOBCYP2A6
SCHEMBL9541503 0.67 TSHR (0.42) NFE2L2TSHRMAOBCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5134240-A Malaria therapy HOFFMANN-LAROCHE, INC. (US) 1992-07-28 US disclosed
US-4977184-A Bicyclic peroxides compositions for and treatment of malaria therewith HOFFMANN-LA ROCHE INC. (US) 1990-12-11 US disclosed