SCHEMBL9735643

SCHEMBL9735643

Fc1c(F)c(F)c(C=P(c2ccccc2)(c2ccccc2)c2ccccc2)c(F)c1F

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.33
CA2 P00918 1/20 0.31
CA4 P22748 1/20 0.31
CA5A P35218 1/20 0.31
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30
NFE2L2 Q16236 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9735648 0.72 NFE2L2 (0.34) HSP90AA1TSHRNFE2L2
SCHEMBL9541494 0.71 NFE2L2 (0.52) ALOX15TSHRNFE2L2
SCHEMBL1132385 0.70 ALDH1A1 (0.39) HSP90AA1CA2CA4CA5AALOX15
SCHEMBL7633171 0.67 HSP90AA1 (0.39) HSP90AA1CA2CA4CA5AALOX15
SCHEMBL9539397 0.64 ALDH1A1 (0.41) HSP90AA1
SCHEMBL16338690 0.64 NFE2L2 (0.43) ALOX15TSHRNFE2L2
SCHEMBL9709624 0.63 CYP11B2 (0.57)
SCHEMBL9539528 0.63 ALDH1A1 (0.48) TSHR
SCHEMBL24193844 0.62 ESR1 (0.50) HSP90AA1CA2CA4CA5ANFE2L2
SCHEMBL9538596 0.62 LMNA (0.42) TSHRNFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5134240-A Malaria therapy HOFFMANN-LAROCHE, INC. (US) 1992-07-28 US disclosed
US-4977184-A Bicyclic peroxides compositions for and treatment of malaria therewith HOFFMANN-LA ROCHE INC. (US) 1990-12-11 US disclosed