SCHEMBL9736741

SCHEMBL9736741

O=C1NC(=O)c2c1c(-c1ccccc1)c(-c1ccccc1)c(P(=O)(O)O)c2P(=O)(O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
WEE1 P30291 9/20 0.43
CHEK1 O14757 8/20 0.43
ADK P55263 1/20 0.39
MAPT P10636 3/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
PTGS2 P35354 2/20 0.37
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA5A P35218 1/20 0.36
MEN1 O00255 2/20 0.36
PRKD3 O94806 2/20 0.36
PRKCG P05129 2/20 0.36
PRKCB P05771 2/20 0.36
CDK4 P11802 2/20 0.36
PRKCA P17252 2/20 0.36
PRKCH P24723 2/20 0.36
PRKCI P41743 2/20 0.36
PRKCE Q02156 2/20 0.36
KMT2A Q03164 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7766596 0.81 MAPT (0.55) WEE1CHEK1ADKMAPTLMNA
SCHEMBL21246791 0.71 MAOA (0.45) WEE1CHEK1ADKMAPTLMNA
SCHEMBL15431517 0.68 CA2 (0.43) MAPTLMNAHTTCA2CA4
SCHEMBL28677769 0.67 GPR84 (0.42) MAPTLMNAHTTCA2CA4
SCHEMBL30753519 0.66 CHEK1 (0.52) WEE1CHEK1ADKMAPTLMNA
SCHEMBL9285018 0.66 ESR1 (0.42) MAPTLMNAHTTPTGS2CA2
SCHEMBL18892992 0.65 HTT (0.44) CHEK1MAPTLMNAHTTMEN1
SCHEMBL6422263 0.63 KDM4E (0.54) ADKMAPTLMNAHTTPTGS2
Phosphoric Acid SCHEMBL5679956 0.63 PDE4A (0.45) MAPTLMNAHTTCA2CA4
Phosphoric Acid SCHEMBL1199529 0.63 PDE4A (0.45) MAPTLMNAHTTCA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5138050-A 6-amido-1-methyl carbapenems MERCK & CO., INC. (US) 1992-08-11 US disclosed
WO-1990000170-A1 NOVEL 6-AMIDO-1-METHYLCARBAPENEMS MERCK & CO., INC. (US) 1990-01-11 WO disclosed
EP-0350211-A2 Novel 6-amido-1-methyl carbapenems MERCK & CO. INC. (US) 1990-01-10 EP disclosed