SCHEMBL9738190

SCHEMBL9738190

Cc1c2n(c3ccc(C(C)C)cc13)CCC2NO

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAD52 P43351 1/20 0.33
PTGES2 Q9H7Z7 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
HSD17B10 Q99714 3/20 0.31
KDM4E B2RXH2 3/20 0.31
CYP1A2 P05177 2/20 0.31
CYP2D6 P10635 2/20 0.31
PAX8 Q06710 1/20 0.31
HTR1D P28221 1/20 0.31
HTR1B P28222 1/20 0.31
TRPA1 O75762 1/20 0.30
PTGS1 P23219 1/20 0.30
CACNA1C Q13936 1/20 0.30
GAA P10253 1/20 0.30
TP53 P04637 1/20 0.30
CYP3A4 P08684 1/20 0.30
HTR1A P08908 1/20 0.30
ADRA2A P08913 1/20 0.30
CHRM1 P11229 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9737169 0.74 ALOX5 (0.34) PTGES2MEN1KMT2AHSD17B10KDM4E
SCHEMBL9736655 0.65 KDM4E (0.37) PTGES2MEN1KMT2AHSD17B10KDM4E
SCHEMBL9737883 0.65 KDM4E (0.63) PTGES2MEN1KMT2AKDM4ETRPA1
SCHEMBL15341790 0.58 CNR1 (0.44) CYP1A2
SCHEMBL8687445 0.58 PTGES2 (0.43) PTGES2MEN1KMT2AKDM4ETRPA1
SCHEMBL25765617 0.58 MEN1 (0.45) MEN1KMT2ATRPA1PTGS1CACNA1C
SCHEMBL12083594 0.58 RORA (0.46) MEN1KMT2AHSD17B10KDM4EHTR1D
SCHEMBL15341787 0.58 CNR1 (0.46)
SCHEMBL26398797 0.57 RORA (0.42) HTR1DHTR1BTRPA1PTGS1CACNA1C
SCHEMBL24667912 0.56 BCHE (0.45) MEN1KMT2AHSD17B10KDM4ETRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992021678-A1 LIPOXYGENASE INHIBITING PYRROLO [1,2a]INDOLE COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1992-12-10 WO disclosed