SCHEMBL9742140

SCHEMBL9742140

COc1cccc(C23CCCN2C(=O)c2ccccc23)c1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 4/20 0.49
PARP1 P09874 3/20 0.47
KMT2A Q03164 1/20 0.43
SLC6A4 P31645 2/20 0.41
SLC6A9 P48067 1/20 0.41
SIGMAR1 Q99720 2/20 0.41
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
OPRL1 P41146 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A3 Q01959 1/20 0.40
BACE1 P56817 1/20 0.40
BACE2 Q9Y5Z0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9740223 0.86 CHRM5 (0.48) CHRM5PARP1SLC6A4SLC6A2SLC6A3
SCHEMBL9742640 0.86 CHRM5 (0.46) CHRM5PARP1KMT2ASLC6A4SLC6A9
SCHEMBL9742113 0.86 CHRM5 (0.43) CHRM5PARP1KMT2ASLC6A4SIGMAR1
SCHEMBL9744849 0.84 PARP1 (0.46) PARP1SIGMAR1
SCHEMBL9743611 0.84 PARP1 (0.46) CHRM5PARP1KMT2ASIGMAR1
SCHEMBL9739723 0.84 LMNA (0.46) CHRM5PARP1KMT2AOPRM1OPRD1
SCHEMBL9740279 0.81 HTT (0.47) CHRM5KMT2A
SCHEMBL9739787 0.81 CHRM5 (0.43) CHRM5KMT2ASLC6A9OPRM1OPRD1
SCHEMBL9740111 0.80 SLC6A2 (0.43) CHRM5KMT2ASLC6A4OPRM1SLC6A2
SCHEMBL9739810 0.79 PARP1 (0.47) CHRM5PARP1SIGMAR1OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992016529-A1 NOVEL ISOINDOLE DERIVATIVES AND MEDICAMENTS CONTAINING THEM BOEHRINGER MANNHEIM GMBH (DE) 1992-10-01 WO disclosed