SCHEMBL9739810

SCHEMBL9739810

COc1ccccc1C12CCCN1C(=O)c1ccccc12

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.47
CHRM5 P08912 5/20 0.44
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
TSHR P16473 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA1A P35348 1/20 0.42
NPY5R Q15761 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
OPRL1 P41146 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
NPC1 O15118 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9738757 0.82 NPC1 (0.43) PARP1CHRM5NPY5ROPRM1SIGMAR1
SCHEMBL9740223 0.82 CHRM5 (0.48) PARP1CHRM5CYP3A4TSHRNPC1
SCHEMBL9740491 0.80 MEN1 (0.40) CHRM5CYP1A2CYP3A4NPC1POLB
SCHEMBL9738947 0.79 HTT (0.42) CHRM5NPY5ROPRM1OPRK1NPC1
SCHEMBL9742140 0.79 CHRM5 (0.49) PARP1CHRM5OPRM1OPRD1OPRK1
SCHEMBL9738938 0.78 NPC1 (0.40) PARP1CHRM5CYP1A2CYP3A4NPY5R
SCHEMBL9738615 0.77 CHRM5 (0.46) CHRM5CYP1A2CYP3A4NPC1POLB
SCHEMBL9739497 0.77 MAPT (0.46) PARP1CHRM5NPC1POLB
SCHEMBL9739249 0.77 SLC6A3 (0.40) PARP1NPC1POLB
SCHEMBL29795000 0.76 LMNA (0.38) CYP1A2CYP3A4TSHRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992016529-A1 NOVEL ISOINDOLE DERIVATIVES AND MEDICAMENTS CONTAINING THEM BOEHRINGER MANNHEIM GMBH (DE) 1992-10-01 WO disclosed