SCHEMBL9749758

SCHEMBL9749758

COC(C)OC.O=Cc1cccc(F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.48
MAOB P27338 2/20 0.48
NFE2L2 Q16236 9/20 0.47
RELA Q04206 1/20 0.46
PTGS1 P23219 2/20 0.45
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
PKM P14618 1/20 0.43
MAPK1 P28482 1/20 0.43
THPO P40225 1/20 0.43
NPC1 O15118 1/20 0.43
CHRM5 P08912 1/20 0.43
GRM5 P41594 1/20 0.43
RAB9A P51151 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
PTGS2 P35354 1/20 0.42
FBP1 P09467 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Isophthalic Dicarboxaldehyde SCHEMBL3536987 0.87 ALDH1A1 (0.47) MAOAMAOBNPC1RAB9AALDH1A1
SCHEMBL24197 0.83
SCHEMBL1574019 0.83 NFE2L2 (0.65) MAOAMAOBNFE2L2PTGS1CYP1A2
SCHEMBL29359478 0.83
SCHEMBL18472616 0.83
Ammonia Solution, Strong SCHEMBL27509053 0.81 NFE2L2 (0.62) MAOAMAOBNFE2L2PTGS1CYP1A2
Hydrochloric Acid SCHEMBL29084496 0.81 NFE2L2 (0.62) MAOAMAOBNFE2L2PTGS1CYP1A2
Hydrochloric Acid SCHEMBL29768617 0.81 NFE2L2 (0.62) MAOAMAOBNFE2L2PTGS1CYP1A2
SCHEMBL10863616 0.81 MAOA (0.49) MAOAMAOBRELAPTGS1NPC1
SCHEMBL8458900 0.79 NPC1 (0.55) MAOAMAOBNFE2L2RELANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0219852-B1 CHARTREUSIN DERIVATIVES, SALTS THEREOF, ANTITUMOROUS COMPOSITIONS CONTAINING THE SAME, AND PROCESSES FOR PRODUCING THE SAME ISHIHARA SANGYO KAISHA, LTD. (JP) 1992-02-05 EP disclosed
US-5064945-A Antitumor Agents ISHIHARA SANGYO KAISHA, LTD. (JP) 1991-11-12 US disclosed
US-4927919-A ANTITUMOR AGENTS ISHIHARA SANGYO KAISHA, LTD. (JP) 1990-05-22 US disclosed
EP-0159708-B1 CHARTREUSIN DERIVATIVES, SALTS THEREOF, ANTITUMOROUS COMPOSITIONS CONTAINING THE SAME, AND PROCESSES FOR PRODUING THE SAME ISHIHARA SANGYO KAISHA, LTD. (JP) 1989-12-13 EP disclosed
US-4760136-A Chartreusin derivatives and salts thereof ISHIHARA SANGYO KAISHA, LTD. (JP) 1988-07-26 US disclosed
EP-0219852-A2 Chartreusin derivatives, salts thereof, antitumorous compositions containing the same, and processes for producing the same ISHIHARA SANGYO KAISHA, LTD. (JP) 1987-04-29 EP disclosed
EP-0159708-A2 Chartreusin derivatives, salts thereof, antitumorous compositions containing the same, and processes for produing the same ISHIHARA SANGYO KAISHA, LTD. (JP) 1985-10-30 EP disclosed